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(furan-2-ylmethyl)({[4-(pyrimidin-2-yloxy)phenyl]methyl})(thiophen-3-ylmethyl)amine
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-(2,2,2-trifluoroethyl)propanamide
4-methoxy-N-{[1-(pyrazin-2-yl)piperidin-3-yl]methyl}benzene-1-sulfonamide
3-(4-fluorophenoxymethyl)-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
4-[4-({4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]-2-methylbut-3-yn-2-ol
N-ethyl-2-[2-(trifluoromethyl)morpholin-4-yl]pyrimidin-4-amine
5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-N-(2-methoxyethyl)pyridin-2-amine
(4aS,8aR)-6-(1H-imidazol-4-ylmethyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
2-[3-(4-fluorophenyl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(phenylsulfanyl)ethan-1-one
N-methyl-4-{4-[1-(methylamino)propyl]phenyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]-4-phenylpiperidine-4-carbonitrile
[(6-ethoxyquinolin-2-yl)methyl](methyl)(1,2-oxazol-3-ylmethyl)amine
[1-methyl-5-(2-phenoxyethyl)-1H-1,2,4-triazol-3-yl](phenyl)methanol
2-(4-fluorophenyl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]acetamide
N-methyl-3-[N-methyl-1-(2-methyl-4-phenyl-1,3-thiazol-5-yl)formamido]butanamide
N,N-dimethyl-2-(pyridine-3-sulfonamidomethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-(3-methoxypropyl)-9-({4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(4-methyl-1,4-diazepan-1-yl)acetamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-6-(2-methoxyphenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(2-ethoxyethyl)-3-methyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H-pyrazole-5-carboxamide
N,N-diethyl-1-[1-(2-ethylbutyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
2-{4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
2-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-oxoethyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
5-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-phenyl-1H-imidazole
2-(2-butyl-1H-imidazol-4-yl)-1-{imidazo[1,2-a]pyridin-2-ylmethyl}-1H-imidazole
N-cyclopropyl-2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-(thiophen-3-ylmethyl)acetamide
(2S,4S)-4-{[(2,5-dimethylphenyl)methyl]amino}-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-{5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]thiophen-2-yl}ethan-1-one
3,5-dimethoxy-N-({1-[3-(methylsulfanyl)propanoyl]piperidin-3-yl}methyl)benzamide
N-(3-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}propyl)-N,5-dimethyl-1,3-oxazole-4-carboxamide
6-(4-methanesulfonylphenyl)-1H-1,3-benzodiazole
1-{[5-(1-benzoylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}-4-methylpiperazine
4,6-dimethyl-2-(propan-2-yl)-5-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methoxy}pyrimidine
N-[2-(1-benzylpiperidin-4-yl)ethyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2-(3-methyl-1,2-oxazol-5-yl)acetamide
1-(2-methyl-4-{[2-(pyridin-2-ylsulfanyl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
2-(5-{3-fluoro-5-methylimidazo[1,2-a]pyridin-2-yl}-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl)pyridine
1-({6-[3-fluoro-5-(propan-2-yloxy)phenyl]pyridin-3-yl}methyl)-4-methylpiperazine
2-[4-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
1-{4-[(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]thiophen-2-yl}ethan-1-one
(3S)-3-({[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)azepan-2-one
1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(1H-imidazol-1-yl)ethan-1-one
N-[(1-benzylpiperidin-3-yl)methyl]-4-methylpyrimidin-2-amine
(1S,5R)-6-benzyl-3-(thiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-(piperidine-1-carbonyl)piperidine-1-carboxamide
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-[(1-benzothiophen-2-ylmethyl)amino]-5-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-{[3-methyl-7-(5-methylthiophene-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenoxypropanamide