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N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylcyclopropanesulfonamide
ethyl 1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
(1S,5R)-3-methyl-6-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
{3-ethyl-1-[1-(pyridine-3-carbonyl)piperidin-4-yl]piperidin-3-yl}methanol
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-1,2,5-thiadiazole-3-carboxamide
3-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
(1S,5R)-3-benzyl-6-[(4-methyl-1,3-thiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-(5-amino-1,3,4-thiadiazol-2-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]ethan-1-one
2-(2,3-difluorophenoxymethyl)-4-(pyrrolidine-1-carbonyl)-1,3-oxazole
2-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-(4-ethylpiperazin-1-yl)-3-(2-methoxy-4-{[(2-phenylethyl)amino]methyl}phenoxy)propan-2-ol
3,6,7-trimethyl-N-(oxan-4-ylmethyl)-1-benzofuran-2-carboxamide
4-cyclopropanecarbonyl-7-(2,6-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1S,5R)-6-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-cyclobutanecarbonyl-1'-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethan-1-one
2-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-1,4-dihydroquinolin-4-one
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1-[2-(trifluoromethyl)phenyl]urea
ethyl 6-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyridine-2-carboxylate
8-[(5-methoxy-2-methyl-3-phenyl-1-benzofuran-6-yl)methyl]-1-methyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[4-(adamantan-1-yl)piperazin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-(azocan-1-yl)-3-(5-methoxy-2-{[(oxan-4-ylmethyl)amino]methyl}phenoxy)propan-2-ol
N-[(3R,4S)-4-cyclopropyl-1-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]pyrrolidin-3-yl]methanesulfonamide
11-[(2-methylpropyl)amino]-4-{[3-(trifluoromethyl)phenyl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
methyl 2-[(1-benzoylpiperidin-4-yl)amino]-2-(3-methylphenyl)acetate
1-[(3,4-dimethylphenyl)methyl]-4-[2-(morpholin-3-yl)acetyl]piperazin-2-one
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)(1,2-oxazol-3-ylmethyl)amine
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
1-ethyl-5-(piperidin-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
6-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
3-{[(5-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}furan-2-yl)methyl]sulfanyl}-4H-1,2,4-triazole
2-cyclopentyl-8-(2,3-dihydroxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(2-chlorophenyl)methyl]-3-methyl-N-(propan-2-yl)pyridine-2-carboxamide
(1R,3S)-3-{[2-(4-fluorophenyl)ethyl](pyridin-3-ylmethyl)carbamoyl}cyclopentane-1-carboxylic acid
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
4-[(4-methoxyphenyl)methyl]-1-(4-phenylbenzoyl)-1,4-diazepan-5-one
1-{1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]piperidin-3-yl}pyrrolidin-2-one
N-{[2-(4-chlorophenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-(thiophen-3-yl)acetamide
(3S,9aR)-3-(4-aminobutyl)-8-(3-phenylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(2,6-difluoro-3-methoxyphenyl)methyl]-3-(methoxymethyl)pyrrolidine
1-(3-chlorophenyl)-4-(1-propylpiperidin-4-yl)piperazine
4,5-dichloro-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}thiophene-2-sulfonamide
1-benzyl-N,5-bis(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-{[2-(methoxymethyl)piperidin-1-yl]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylic acid
N-[(1-ethyl-1H-indazol-3-yl)methyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
2-{1-[1-(3-methylquinolin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[3-(morpholine-4-carbonyl)piperidin-1-yl]propan-1-one
3-{1-[2-(2-phenyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N,N-dimethyl-4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
N-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-4-(pyrrolidine-1-sulfonyl)piperazine-1-carboxamide