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N-cyclopropyl-1-[1-(1,3-thiazol-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(2S)-2-amino-1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(1H-imidazol-4-yl)propan-1-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[(4aS,7aR)-4-(2-methylpropyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxo-N-phenylacetamide
1-(2-{[(2-fluorophenyl)methyl](methyl)amino}ethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
6,7-dimethoxy-3-[(3,4,5-trifluorophenyl)methyl]-3,4-dihydroquinazolin-4-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
6-(2,3-dimethylquinoxaline-6-carbonyl)-2-(2-hydroxyethyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
1-{3-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-3-oxopropyl}azepan-2-one
1-(propan-2-yl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-pyrazole-4-carboxamide
ethyl 1-[7-chloro-3-({[(1-hydroxycyclohexyl)methyl]amino}methyl)quinolin-2-yl]piperidine-3-carboxylate
2-(1H-pyrazol-1-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
2-fluoro-N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-5-sulfamoylbenzamide
[2-(2,5-dimethylphenoxy)ethyl](methyl)(quinoxalin-2-ylmethyl)amine
3-chloro-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}thiophene-2-carboxamide
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-1H-1,2,3-benzotriazole-5-carboxamide
1-(4-{[4-(cyclopentyloxy)phenyl]methyl}-6-hydroxy-1,4-diazepan-1-yl)ethan-1-one
dimethyl[1-(3-{[4-(thian-4-yl)piperazin-1-yl]methyl}phenyl)ethyl]amine
6-[2-(benzyloxy)ethyl]-N,N-dimethylpyrimidin-4-amine
1-[(2-chloro-6-fluorophenyl)methyl]-3-cyclopropyl-5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
N-[2-(4-fluorobenzenesulfonyl)ethyl]-1-(propan-2-yl)-1H-pyrazole-3-carboxamide
2-methyl-7-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-(2-{[2-(dimethylamino)ethyl]amino}pyrimidin-4-yl)-2-ethoxybenzoic acid
(4aR,7aS)-1-(cyclopropylmethyl)-4-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1H-imidazol-2-ylmethyl)-3-(2-oxoazepan-1-yl)propanamide
1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3-[2-(2-methylphenyl)ethyl]piperidine
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
N-(2-ethyl-3-methyl-1-benzofuran-7-yl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
2-methyl-4-[3-(2-methyl-4-phenylpiperazine-1-carbonyl)phenyl]butan-2-ol
4-{4-[(4-methoxyphenyl)methyl]piperazin-1-yl}-2-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-(2H-1,3-benzodioxol-5-yl)-5-[(2,3-dihydro-1,4-benzodioxin-5-yloxy)methyl]-1,2,4-oxadiazole
1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-3-(3-methoxyphenyl)propan-1-one
1-{1-[3-(dimethylamino)pyrazin-2-yl]piperidin-4-yl}piperidin-4-ol
5-fluoro-N4-methyl-N2-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrimidine-2,4-diamine
1'-(1-benzothiophene-2-carbonyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[3,5-dimethyl-4-(naphthalene-1-sulfonamido)-1H-pyrazol-1-yl]acetic acid
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(2-methyl-1-benzofuran-5-carbonyl)pyrrolidin-3-yl]methanol
2-[N-(3-fluorophenyl)methanesulfonamido]-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[3-(2-methoxyacetamido)-2-methylphenyl]azetidine-1-carboxamide
1-(4-aminopyrimidin-2-yl)-4-(3-tert-butyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-{4-[4-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}pyridine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,2-dimethyl-1H-1,3-benzodiazole-5-carboxamide
N-[1-(7-methoxy-4-methylquinazolin-2-yl)pyrrolidin-3-yl]-N-methylacetamide
N-[1-(cyclohexylcarbamoyl)piperidin-4-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
9-benzoyl-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-4-amino-1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}piperidin-3-ol
8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-3,3-diphenylpropan-1-one
N-(4-{[(butan-2-yl)(cyclopentyl)amino]methyl}phenyl)acetamide
N-[(3-chloro-4-fluorophenyl)methyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide