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1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
1-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4-(4H-1,2,4-triazol-4-yl)benzamide
2-(cyclopent-2-en-1-yl)-1-{6-methyl-5-[5-(1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}ethan-1-one
4-hydroxy-1-[8-(trifluoromethyl)quinolin-4-yl]piperidine-4-carboxylic acid
2-(1-benzyl-4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
N-({4-hydroxy-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]azepan-4-yl}methyl)benzamide
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-bromobenzamide
2-chloro-4-({[1-(4-methyl-1H-imidazol-2-yl)propyl]carbamoyl}amino)-N-(propan-2-yl)benzamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
N-butyl-N-[(3-methylthiophen-2-yl)methyl]-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
2-(morpholin-4-yl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-2-(pyridin-3-yl)acetamide
2-{2-[4-(oxolan-2-ylmethyl)piperazin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
1-({4-methyl-5-[1-(propan-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
2-(2-methoxyethyl)-9-[5-(propan-2-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
4-[(3-methylphenyl)methyl]-3-(1-methylpiperidin-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]pyridine-4-carbonitrile
N-methyl-6-oxo-1-(3-phenylpropyl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)piperidine-3-carboxamide
5-[1-(1,4-dioxan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]-2-propylpyrimidine
N-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-N-methyl-1-(3-phenylpropyl)piperidin-3-amine
1-(2-methanesulfonylethyl)-2-(3-methylthiophen-2-yl)-1H-imidazole
N-[(2-methoxyphenyl)methyl]-5-methyl-6-(4-methylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
2-[methyl({4-methyl-5-[1-(2-methylpyridin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
8-(2-aminoacetyl)-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-(pyrrolidin-1-yl)pyrimidin-2-amine
3-(4-hydroxyphenyl)-N-[(2S)-1-methoxy-3-phenylpropan-2-yl]-1H-pyrazole-5-carboxamide
5-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
ethyl 3-({4-[2-(phenylcarbamoyl)ethyl]piperidine-1-carbonyl}amino)propanoate
2-{2-methyl-2,8-diazaspiro[4.5]decane-8-carbonyl}benzonitrile
N-(3-chloro-4-methoxyphenyl)-3-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-yl]propanamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]furan-2-carboxamide
3-hexyl-8-[(1-methyl-1H-imidazol-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[1-(9H-fluoren-2-ylmethyl)piperidin-4-yl]-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
3-[(3-hydroxyazetidin-1-yl)sulfonyl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
4-(4-ethoxybenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
N-[(2-methoxyphenyl)methyl]-2,6-dioxo-N-(pyridin-3-ylmethyl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
methyl 2-(1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
3-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-6-(propan-2-yl)-1,2-dihydropyridin-2-one
2-{2-[2-(dimethylamino)phenyl]-4-methylphenoxy}acetamide
{[4-(methylsulfanyl)phenyl]methyl}[(2-phenoxypyridin-3-yl)methyl]amine
N-(furan-3-ylmethyl)-N-methyl-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-[2-(adamantan-1-yl)-4-hydroxypyrimidine-5-carbonyl]-2-methyl-1,4-diazepan-5-one
1-[3-(2-methylpropyl)-1,2-oxazole-5-amido]-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
3-{5-[2-(methylamino)-1,3-thiazole-4-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
{2-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-1,3-thiazol-4-yl}methanol
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-2-(pyridin-4-ylsulfanyl)acetamide
N-{[1-(4-chlorophenyl)cyclopropyl]methyl}-2-(dimethylamino)-2-(2-fluorophenyl)acetamide