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N-({1-[(3-chloro-1-benzothiophen-2-yl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
(2R,3R)-1'-(1,2,5-oxadiazole-3-carbonyl)-3-(1,2,3,6-tetrahydropyridin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(cyclohexylmethyl)-4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidine
1-(3-chloro-2-propoxyphenyl)-3-methylurea
1-(2,2-dimethylpropyl)-3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
1-{furo[3,2-c]pyridin-4-yl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
2-(dimethyl-1,3-thiazol-4-yl)-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}acetamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-3-ethoxy-4-(prop-2-en-1-yloxy)benzamide
1-(4-fluorophenyl)-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
6-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-N-propylpyridine-3-carboxamide
4-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-2-(prop-2-en-1-yl)phenol
2-{[4-(1H-pyrazol-3-yl)phenyl]methoxy}ethan-1-amine
5-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-4,6-dimethyl-1,2,3,4-tetrahydropyrimidin-2-one
3-methyl-7-(5-propylthiophene-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-methyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]pyrido[2,3-d]pyrimidin-4-amine
1-{[2-(cyclopentyloxy)phenyl]methyl}-4-(2-methanesulfonylethyl)piperazine
8-{[2-(difluoromethoxy)phenyl]methyl}-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N3-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-N1-(pyridin-3-yl)propane-1,3-diamine
N-(2-{[1-(3-methoxyphenyl)propan-2-yl]amino}ethyl)-N-methylmethanesulfonamide
N-[3-(4-{[(3S)-2-oxoazepan-3-yl]amino}piperidin-1-yl)phenyl]-4-phenylbutanamide
5-(1-butylpyrrolidin-2-yl)-N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]thiophene-2-carboxamide
3-chloro-N-cyclopentyl-4-({1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}oxy)benzamide
N-[2-(3-methoxyphenyl)ethyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-hydroxy-1-(2-methoxyethyl)-3-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-ylmethyl)piperidin-2-one
2-{cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}-2-(4-fluoro-3-methylphenyl)acetic acid
N-(4-{1-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide
3-[2-(dimethylamino)ethyl]-8-(1H-indole-6-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-cyclopropyl-2-phenyl-N-(pyridin-3-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
7-{[3-(benzyloxy)phenyl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
(3aR,6aR)-2-methanesulfonyl-5-[(5-methylthiophen-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
N-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}benzamide
2-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}benzoic acid
N-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-1-(methoxymethyl)cyclobutane-1-carboxamide
1-ethyl-3-(morpholine-4-carbonyl)-N-{[3-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(2-hydroxypropyl)-9-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(butan-2-yl)-2-[methyl(pyridin-4-ylmethyl)amino]-N-(thiophen-3-ylmethyl)acetamide
1-(1H-imidazol-2-ylmethyl)-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
(1S,5R)-3-benzyl-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[7-(2,6-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
ethyl 1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylate
6-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}pyridine-3-carboxylic acid
2-methyl-8-(2-methyl-1,3-benzothiazole-6-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-({1-[(4-chlorophenyl)methyl]piperidin-4-yl}oxy)-N-cyclopropyl-4-methoxybenzamide
N-[2-(ethylsulfanyl)phenyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carboxamide
5-(3-ethyl-4-methyl-1H-pyrazol-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
11-methyl-4-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-(5-chloro-2-methoxyphenyl)-3-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]propanamide
4-methyl-5-[3-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,3-oxazole
2-methyl-4-(1-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-1,3-thiazole