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3-(1H-indazol-3-yl)benzoic acid
1-[4-(morpholin-4-yl)-3-[3-(1H-pyrazol-1-yl)phenyl]phenyl]ethan-1-one
1-[2-(4-phenylphenyl)acetyl]-4-(pyridin-3-ylmethyl)-1,4-diazepan-5-one
N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-1-ethyl-1H-pyrazole-3-carboxamide
methyl 3-{methyl[2-(4-methylpiperidin-1-yl)ethyl]carbamoyl}benzoate
4-{[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]methyl}benzonitrile
2-[3-(3-{7-methylthieno[3,2-d]pyrimidin-4-yl}phenyl)-1H-pyrazol-1-yl]ethan-1-ol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(pyridin-4-yl)quinoline-4-carboxamide
(4-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1,4-oxazepan-6-yl)methanol
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
2-[2-(3-hydroxyphenyl)ethyl]-N-(1H-indazol-7-yl)piperidine-1-carboxamide
methyl(quinolin-6-ylmethyl)[(4-{[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
3-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1-[2-(prop-2-en-1-yloxy)phenyl]urea
6-methyl-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]pyridine-2-carboxamide
2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-[2-(methylsulfanyl)phenyl]acetic acid
(2E)-3-(2-chlorophenyl)-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(propan-2-yloxy)phenyl]methyl}prop-2-enamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
1-[2-(1,3-dihydro-2-benzofuran-5-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[(2-methoxyphenyl)methyl]piperidine-3-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4H-thieno[3,2-b]pyrrole-5-carboxamide
3-(3-methoxyphenyl)-N-[1-(3-methylphenyl)piperidin-4-yl]-1H-pyrazole-5-carboxamide
1-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
methyl (2S)-1-(3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanoyl)pyrrolidine-2-carboxylate
1-[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
(4aS,8aR)-6-[2-(2-methoxyphenyl)acetyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-[(3R,4R)-1-[(4-cyano-5-methyl-1H-pyrrol-2-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-(pyridin-2-yl)piperidine-3-carboxamide
methyl 2-(1H-imidazol-2-yl)-3,5-dimethoxybenzoate
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-[1-(pyridin-3-ylmethyl)piperidin-3-yl]propanamide
3-(1H-1,3-benzodiazol-1-yl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
[2-(dimethylamino)ethyl](ethyl)({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
4-[(4-cyclopentylpyrimidin-2-yl)amino]-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
2-(propan-2-yl)-1-[2-(thiophen-2-yl)ethyl]-1H-imidazole
2-{4-[(3-fluoro-4-methylphenyl)methyl]piperazin-1-yl}-6-(pyrrolidine-1-carbonyl)pyrazine
3-{[(1S,2R)-2-aminocyclobutyl]sulfamoyl}thiophene-2-carboxylic acid
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
5-fluoro-2-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}-N,N-dimethylpyrimidin-4-amine
1-(2-chlorophenyl)-4-(dimethyl-1,3-oxazole-5-carbonyl)piperazin-2-one
(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-(3-methyl-1H-pyrazole-5-carbonyl)-8-azabicyclo[3.2.1]octane
4-ethyl-6-(4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)pyrimidine
2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-phenylacetic acid
3-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}naphthalen-2-ol
4-ethyl-1-methyl-3-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4S)-1-[2-(1H-indol-3-yl)ethyl]-4-methylpiperidine-3,4-diol
N-[(3R,4S)-1-[3-(methylsulfanyl)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-(2-oxopiperidin-1-yl)acetamide
1-cyclohexyl-3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-(2-hydroxy-2-phenylethyl)urea
N-benzyl-N-methyl-1-(6-methylpyridine-3-carbonyl)piperidin-3-amine
6-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]quinoxaline