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4-[(2S)-1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-2-carbonyl]morpholine
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}propanamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}pyrrolidine-1-carboxamide
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2,5-dimethoxybenzamide
4-chloro-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}benzene-1-sulfonamide
N-(1,3-dihydroxy-2-methylpropan-2-yl)-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[2-(dimethylamino)ethyl]-1-ethyl-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)piperidine-4-carboxamide
1-(1-benzofuran-2-ylmethyl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1,4-diazepan-6-ol
ethyl 3-benzyl-1-[(2-chloro-6-methylphenyl)carbamoyl]piperidine-3-carboxylate
N,N-dimethyl-5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}furan-2-carboxamide
4-hydroxy-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine-3-carboxamide
3-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-cyclopentylurea
methyl 2-(diethylsulfamoyl)-6-(2,6-difluorobenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
9-(6-methoxyhexanoyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(4-chloro-2-{[3-(3-methylphenoxy)azetidin-1-yl]methyl}phenoxy)acetamide
1-methyl-6-(propan-2-yl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[2-(2-fluorophenyl)ethyl]-3-(3-methyl-1,2-oxazol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-3-(1-methylpiperidin-2-yl)propanamide
3-(1H-imidazol-1-ylmethyl)-1-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}piperidine
methyl (2S)-3-(4-hydroxyphenyl)-2-({8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}amino)propanoate
2-({2-[(dicyclopropylmethyl)(methyl)carbamoyl]phenyl}amino)acetic acid
2-benzyl-9-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-ethyl-4-methyl-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}-1H-pyrazole-5-carboxamide
3-{5-[(2,5-dimethoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenol
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chloro-2-methylphenyl)urea
(1-{2-[(6-methoxypyrimidin-4-yl)amino]ethyl}piperidin-2-yl)methanol
(3R,4R)-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
(3R,4R)-4-methyl-3-(propan-2-yl)-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}pyrrolidin-3-ol
1-[3-(morpholine-4-carbonyl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
2-[benzyl(methyl)amino]-N-(2-hydroxypropyl)-2,3-dihydro-1H-indene-2-carboxamide
4-(5-chlorothiophen-2-yl)-N,N-dimethylbenzamide
4-(4-ethyl-1H-pyrazol-5-yl)-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidine
1-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}pentane-1,4-dione
N-({1-[(8-methoxyquinolin-2-yl)methyl]pyrrolidin-3-yl}methyl)cyclopropanecarboxamide
ethyl 3-[(2-methylphenyl)methyl]-1-(2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)piperidine-3-carboxylate
4-{5-[(2E)-but-2-en-1-yl]-1,3,4-oxadiazole-2-carbonyl}-2,2-dimethylmorpholine
5-cyclopropyl-N-{1-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-1,3,4-oxadiazol-2-amine
2-(cyclopropylmethyl)-9-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-2-{[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
(3aR,6aR)-2-(2,5-dimethylbenzoyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-2-fluoro-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
N,N-diethyl-3-[4-(1,3-oxazol-5-yl)phenyl]benzamide
(4aS,8aS)-2-{[4-methoxy-3-(prop-2-en-1-yl)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
3-{5-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}benzonitrile
N-methyl-N-(prop-2-en-1-yl)-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-[(2-methoxyphenyl)methyl]-2-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]acetamide
4-(3-{8-ethyl-2,8-diazaspiro[5.5]undecane-2-carbonyl}phenyl)-2-methylbutan-2-ol
4-[3-(aminomethyl)piperidin-1-yl]-6-ethyl-5-methylpyrimidin-2-amine