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6-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-2-methylpyrimidin-4-amine
5-(3-methylphenyl)-2-(pyridin-4-yl)-4-[1-(thiophene-2-carbonyl)piperidin-4-yl]pyrimidine
1-{7-chloro-3-[(cycloheptylamino)methyl]quinolin-2-yl}piperidin-3-ol
(3S,4S)-1-{[4-(benzyloxy)phenyl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N,N-dimethylacetamide
1-(4-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-(1-benzothiophen-5-ylmethyl)-2-(2-ethyl-1H-imidazol-1-yl)acetamide
5-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
1-cyclopropyl-4-({[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}methyl)pyrrolidin-2-one
5-(1,3-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1H-imidazole
(1S,5R)-6-(3,5-difluoropyridine-2-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N,N-bis(2-hydroxyethyl)-3-[(3S,4R)-1-(pyridin-2-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
N-(4-{4-[(butan-2-yl)amino]piperidin-1-yl}phenyl)-2-fluorobenzamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
[(4aS,8aR)-6-{[5-(2-fluorophenyl)furan-2-yl]methyl}-decahydro-1,6-naphthyridin-4a-yl]methanol
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
(1S,5R)-6-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-3-(pyridin-2-ylmethyl)-6-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
{[(3S,4R)-1-(3-chlorothiophene-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
[(2,4-difluorophenyl)methyl](methyl)[1-(pyrimidin-4-yl)ethyl]amine
2,6-dimethyl-3-[4-(4-methylphenyl)piperazine-1-carbonyl]quinoline
(3aS,6aR)-5-(3,6-dimethylpyrazin-2-yl)-3-[3-(4-methoxyphenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methyl-N-(oxolan-3-yl)thieno[2,3-d]pyrimidine-6-carboxamide
2-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-4-amine
N-(2H-1,3-benzodioxol-5-yl)-7-(3-methoxypropanamido)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-(2-amino-2-methylpropyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-[(pyridin-3-ylmethyl)amino]pyrrolidine-2-carboxamide
4-hydroxy-1-[(4-methylphenyl)carbamoyl]piperidine-4-carboxylic acid
(3R,4R)-1-[3-(1H-pyrazol-1-yl)propyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
3-(3-fluorophenyl)-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
N,2-dimethyl-N-(oxan-2-ylmethyl)-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3-[(4-methanesulfonylmorpholin-2-yl)methyl]-1-[3-(1,3-oxazol-5-yl)phenyl]urea
{1-[2-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]piperidin-2-yl}methanol
8-(pyridin-4-ylmethyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-methyl-8-(1-methyl-1H-pyrazole-5-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[1-(ethanesulfonyl)azepan-3-yl]-5-oxo-5-phenylpentanamide
N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl]propan-1-ol
2-(3-acetyl-1H-indol-1-yl)-1-[3-(pyridin-2-yl)azetidin-1-yl]butan-1-one
N-[phenyl(pyridin-2-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N2,N2,N4,5,6-pentamethyl-N4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]pyrimidine-2,4-diamine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]cyclopropanecarboxamide
N-(1-hydroxybutan-2-yl)-3,5-dimethyl-N-(pyridin-3-ylmethyl)-1H-indole-2-carboxamide
N-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-propyl-1H-pyrazole-4-carboxamide
2-methyl-4-{5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]furan-2-yl}but-3-yn-2-ol
5-(2-methoxyacetamido)-1-(2-phenylethyl)-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}-1H-1,3-benzodiazole-7-carboxamide
1-(cyclopropanesulfonyl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
1-(4-methyl-1,3-thiazole-5-carbonyl)-4-phenoxypiperidine-4-carboxylic acid