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2-(5-methyl-1,2-oxazol-3-yl)-1-{[4-(methylsulfanyl)phenyl]methyl}piperidine
N-benzyl-N,1-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-sulfonamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-4-(2-oxopyrrolidin-1-yl)benzamide
1-(2-methoxybenzoyl)-4-{[4-(pyridin-2-yl)phenyl]methyl}piperazine
4-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-1,2-dimethylpiperazine
1-(1-cyclohexylpiperidine-4-carbonyl)-4-(4H-1,2,4-triazol-3-yl)piperidine
(1S,5R)-6-(cyclopropylmethyl)-3-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-methylpyrazine
3-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
4-{[(3S,5R)-1-[(3,4-dimethoxyphenyl)methyl]-5-(piperidine-1-carbonyl)piperidin-3-yl]methyl}morpholine
methyl 2-(ethylsulfamoyl)-6-[4-(1H-indol-3-yl)butan-2-yl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]propanamide
1-{1-[1-(3-methoxyphenyl)piperidin-4-yl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
(3S,5S)-N-(2,3-dihydro-1H-inden-2-yl)-1-(pyridin-4-ylmethyl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
2-ethyl-5-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidine
N,5-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]benzonitrile
2,6-dimethoxy-3-[6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]pyridine
3-[1-(4-methyl-1H-imidazole-5-carbonyl)azetidin-3-yl]pyridine
3-chloro-2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
N-{[(2S,4S)-1-[3-(1,3-benzothiazol-2-yl)propanoyl]-4-fluoropyrrolidin-2-yl]methyl}-2-methoxyacetamide
N-(1-benzofuran-2-ylmethyl)-1-cyclopentanecarbonylpiperidine-4-carboxamide
8-(2-methoxy-4-methylbenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2S,4R)-4-[2-(dimethylamino)acetamido]-N-ethyl-1-(2-oxo-2-phenylacetyl)pyrrolidine-2-carboxamide
N-[(1S)-1-cyclohexylethyl]-2-methyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
(2R,3R,6R)-5-(2,4-dimethylpyrimidine-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(4-ethoxyphenyl)ethan-1-one
3-[2-(dimethylamino)ethyl]-8-(3-propyl-1H-pyrazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}propanamide
N-cyclopropyl-1-[1-(2,2-dimethylpropanoyl)piperidin-4-yl]piperidine-3-carboxamide
1-(2,3-difluorobenzoyl)-3-(2-ethylphenoxy)azetidine
[(3R,4R)-1-(4-chloro-3-methylbenzoyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
N-[(3S,4R)-1-(2-{[(2-methylphenyl)methyl]sulfanyl}acetyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
9-methyl-6-(pyrimidin-5-yl)-2,3,4,9-tetrahydro-1H-carbazol-1-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(4-methyl-1,4-diazepan-1-yl)propanamide
2-amino-N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}acetamide
2-[5-(1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-1,2,3-triazol-4-yl)furan-2-yl]benzonitrile
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
1-(cyclopropylmethyl)-5-[2-(4-methoxyphenoxy)acetyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-benzyl-6-(2,5-dimethoxyphenyl)-2-(dimethylamino)-N-[2-(dimethylamino)ethyl]pyridine-3-carboxamide
1-(3-methoxypropyl)-8-(2-methylpropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-acetyl-N-[(2-methylphenyl)(thiophen-2-yl)methyl]piperidine-4-carboxamide
N-ethyl-4-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-oxoimidazolidin-1-yl)benzamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,1,2,5-tetramethyl-1H-pyrrole-3-carboxamide
3-(5-chloro-2-methoxypyridin-4-yl)-5,6-dimethyl-1,2-dihydropyridin-2-one
[(3,4-dimethoxyphenyl)methyl](methyl)[(1-methylcyclopropyl)methyl]amine
6-fluoro-4-{3-[(4-fluorophenyl)methoxy]azetidine-1-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
N-{4-chloro-3-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenyl}-2-methoxyacetamide