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(benzylsulfamoyl)(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)amine
4-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
1-(5-methyl-1,2-oxazole-3-carbonyl)-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
methyl 3-[(2-chloro-6-fluorophenyl)methyl]-9-(cyclopentyloxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
8-[(3-fluoro-4-methoxyphenyl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-[(3-fluorophenyl)methyl]-4-[(2-methoxyethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
6-(1,3-benzothiazol-2-ylmethyl)-N-[2-(cyclohex-1-en-1-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]propan-1-one
1-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-6-hydroxy-1,4-diazepan-1-yl]-3-(1H-pyrazol-4-yl)propan-1-one
2,6-dimethyl-5-{2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,3-benzodiazole
4-[4-(1H-imidazol-1-ylmethyl)phenyl]-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
(4-{[1-(1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-chloro-4-fluoro-5-methylphenyl)-4-[2-(dimethylamino)ethoxy]piperidine-1-carboxamide
[4-(5-methyl-2-phenylfuran-3-carbonyl)-1,4-oxazepan-6-yl]methanol
N-[(2-fluorophenyl)methyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-[4-({[1-(pyrimidin-2-yl)piperidin-3-yl]amino}methyl)phenyl]acetamide
2-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-[4-(1-cyano-1-methylethyl)phenyl]-5-(pyrrolidine-1-sulfonyl)benzoic acid
3-ethyl-8-[(4-methoxynaphthalen-1-yl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(3-{[(2-chlorophenyl)methyl]sulfanyl}propyl)imidazo[1,2-a]pyridine-6-carboxamide
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
N-[2-({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}amino)ethyl]pyridine-4-carboxamide
N-{2-[4-phenyl-5-(1,2,3-thiadiazol-4-yl)-1H-imidazol-1-yl]ethyl}aniline
1-(4-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}piperidin-1-yl)ethan-1-one
(3S,4S)-1-[2,4-bis(trifluoromethyl)benzoyl]piperidine-3,4-diol
N-[4-(3-methoxypiperidine-1-carbonyl)phenyl]ethane-1-sulfonamide
N-[3-(3,5-difluoro-4-methoxyphenyl)phenyl]acetamide
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(3-hydroxy-4-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
3-{2-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-1,3-thiazolidine-2,4-dione
(1S,5R)-6-(cyclobutylmethyl)-3-[(4-methoxypyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[2-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)phenyl]-1H-1,2,3,4-tetrazole
4-acetamido-3-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}benzamide
2,3,6-trimethyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-4-carboxamide
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(2-phenyl-1,3-thiazol-4-yl)ethan-1-one
5-(methoxymethyl)-N-{2-[methyl(phenyl)carbamoyl]phenyl}furan-2-carboxamide
4-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridin-1-ium-1-olate
(2S,4S)-4-[(1-benzylpiperidin-4-yl)amino]-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
2-{[2-(1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]methyl}pyridine
N'-[(5-methylthiophen-2-yl)methyl]-N'-(prop-2-en-1-yl)pentanediamide
4-(pyridin-2-yl)-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}pyrimidin-2-amine
4,5-dimethyl-6-(pyridin-3-yl)-2-(trifluoromethyl)pyrimidine
(3R,4R)-1-(1-ethyl-1H-pyrazole-4-carbonyl)-3,4-dimethylpyrrolidin-3-ol
1-(1-methylpiperidin-4-yl)-4-[(5-propylfuran-2-yl)methyl]piperazine
4-[(1-{1-azabicyclo[2.2.2]octan-3-yl}piperidin-4-yl)oxy]-3-chloro-N-(2-methoxyethyl)benzamide
(4-methyl-5-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methanol
(3R,5S)-1-benzyl-N-[(2,4-difluorophenyl)methyl]-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrrolidin-3-amine