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1-[6-(2,3,4-trimethoxyphenyl)pyridin-2-yl]ethan-1-ol
{[4-ethyl-5-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
N-[4-(3-methylphenyl)phenyl]-1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidine-4-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-4-(pyridin-2-yl)piperazine
5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
6-(aminomethyl)-N-methyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}pyrimidin-4-amine
5-{[(3,4-difluorophenyl)methyl]amino}-1-ethyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(2-{methyl[4-(pyridin-2-yl)pyrimidin-2-yl]amino}ethyl)piperidin-2-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)thiophene-2-carboxamide
2-{2-[(1,4-dithiepan-6-yl)amino]ethyl}-1,2-dihydrophthalazin-1-one
(4S)-3,3,4-trimethyl-1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperidin-4-ol
(1R,9aR)-N-{2-[4-(dimethylamino)phenyl]ethyl}-octahydro-1H-quinolizine-1-carboxamide
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2-hydroxy-2-(4-methoxyphenyl)ethan-1-one
4-(6-chloro-1H-1,3-benzodiazol-2-yl)-N-methylbenzene-1-sulfonamide
N-(1-carbamoylcyclopentyl)-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
(1R,5S,6R)-N-(2-hydroxyethyl)-3-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
1-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]butan-2-ol
2-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-3,5-dimethoxybenzoic acid
5-chloro-15-methyl-9-(5-methylthiophen-2-yl)-12-(pyrrolidine-1-carbonyl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
2-acetamido-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylacetamide
[2,4,6-trimethyl-3-({[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]amino}methyl)phenyl]methanol
N-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-(pyridin-3-yl)azetidine-1-carboxamide
3-{[6-(propan-2-yl)pyrimidin-4-yl]amino}-2-(thiophen-3-ylmethyl)propan-1-ol
1-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(pyrrolidin-1-yl)propan-1-one
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(furan-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(1R,5S,6R)-3-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
1-{3-oxo-3-[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propyl}piperidin-2-one
N-ethyl-3-[({[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}carbamoyl)amino]benzamide
1-(3,4-dimethoxybenzenesulfonyl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
5-{[1-(2H-1,3-benzodioxol-5-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
1-amino-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}cyclobutane-1-carboxamide
4-(3-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-8-methylimidazo[1,2-a]pyridine-2-carbonyl)morpholine
2-(2,4-dimethoxyphenyl)-5-(pyrrolidin-1-ylmethyl)pyridine
2-(2,4-dichlorophenoxy)-N-methyl-N-(1,3-thiazol-2-ylmethyl)acetamide
2-(4-{[ethyl(pyridin-3-ylmethyl)amino]methyl}phenyl)-6-(methoxymethyl)-3,4-dihydropyrimidin-4-one
(4aR,7aS)-1-benzyl-4-(1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-4-chloro-3-methyl-1H-pyrazole-5-carboxamide
2-{4-methyl-6-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrimidin-2-yl}phenol
5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-N-cyclohexyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3,3-diethylurea
3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}-3-{[4-(propan-2-yl)piperazin-1-yl]methyl}piperidin-2-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-(propan-2-yl)piperidine-3-carboxamide
(2S,4R)-4-{[(2,5-difluorophenyl)methyl]amino}-N-ethyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
(1-{[1-(7-chloroquinoxalin-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
N-[(3S,5S)-1-cyclopropanecarbonyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]pyridine-4-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-[1-(1H-indole-3-carbonyl)piperidin-3-yl]propanamide
5-[2-(dimethylamino)acetyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid