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(1R,5S,6R)-3-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
(2S)-N,N-dimethyl-1-{4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carbonyl}pyrrolidine-2-carboxamide
N-[(3-methylpyridin-4-yl)methyl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N-[(3S,4R)-1-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidine-3-carboxamide
5-acetyl-N,2,4-trimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-pyrrole-3-carboxamide
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclohexyl-4-[4-(1H-pyrazol-4-yl)butanamido]piperidine-1-carboxamide
3-{[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]sulfonyl}pyridine
4-(1H-imidazol-2-yl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-[1-(furan-2-ylmethyl)-4-(1H-indole-6-carbonyl)piperazin-2-yl]ethan-1-ol
2-amino-4-[4-hydroxy-3-methoxy-5-(prop-2-en-1-yl)phenyl]-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
3-[(1-{2-[cyclopentyl(methyl)amino]acetyl}pyrrolidin-3-yl)methyl]benzamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-(3-fluorophenyl)-3-{1-[1-(2-hydroxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
methyl 6-benzoyl-2-[(3,5-dimethylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-amino-N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(propan-2-yl)pyrimidine-4-carboxamide
1-(3-ethyl-1H-pyrazole-4-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(5-propylpyrimidin-4-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[4-(2-phenoxyethyl)piperazine-1-carbonyl]pyridin-2-amine
(1S,6R)-9-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-({[2-(cyclohex-1-en-1-yl)ethyl]amino}methyl)-4-(pyrazin-2-yl)phenol
1-(1H-1,2,3-benzotriazol-5-yl)-3-(2-methoxyethyl)-3-propylurea
3-{[ethyl(pentan-3-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-(2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-oxoethyl)-4H,5H,6H,7H,8H,9H-[1,2,4]triazolo[3,2-b]quinazolin-9-one
N-[(1S,2R)-2-{[1-(3-methylphenyl)piperidin-4-yl]amino}cyclobutyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(2S)-2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]propan-1-one
1-[9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
3-(2-fluorophenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
2-{[1-(dimethylamino)hex-5-en-2-yl]oxy}-N-ethylpyridine-4-carboxamide
4-(4-cyclopropyl-4H-1,2,4-triazol-3-yl)-2-methoxyphenol
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(2,3-dihydro-1-benzofuran-5-carbonyl)piperidine
N-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carboxamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(furan-3-ylmethyl)piperazin-2-yl}ethan-1-ol
[(2R)-1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]pyrrolidin-2-yl]methanol
2-amino-N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-butyl-3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidine-1-carboxamide
4-{[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-4-ylmethyl)benzamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-methylpiperidine-4-carboxamide
N-ethyl-3-(3-hydroxy-3-methylbutyl)-N-(pyridin-3-ylmethyl)benzamide
2-(4-fluorophenoxymethyl)-4-hydroxy-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)pyrimidine-5-carboxamide
5-(2-methoxyquinolin-3-yl)-N-methylfuran-2-carboxamide
2-phenyl-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-[(2,4-dimethoxyphenyl)methyl]-3-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-2-one
N-{1-[(2,3,4-trimethoxyphenyl)methyl]-1H-pyrazol-5-yl}morpholine-4-carboxamide