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(3S,4R)-4-(2-methoxyphenyl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidine-3-carboxylic acid
(3aR,6aR)-2-acetyl-5-(4-ethyl-5-methylpyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-7-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
1-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]-2-(propan-2-yloxy)ethan-1-one
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
3-[2-(3,4-difluorophenyl)ethyl]-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
N-{1-oxaspiro[4.4]nonan-3-yl}-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butanamide
(3aR,6aR)-2-(4-chlorobenzoyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-({[4-methyl-7-(methylsulfanyl)quinolin-2-yl]amino}methyl)-1λ6-thiolane-1,1-dione
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(methylsulfanyl)ethan-1-one
(3aR,6aR)-2-(3-chlorobenzoyl)-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-butyl-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-imidazole
4-[2-(aminomethyl)morpholin-4-yl]-N-(2-methoxyethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-4-hydroxy-4-phenylpiperidine-1-carboxamide
N-cyclopentyl-4-{2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}-4-oxobutanamide
1-(2-{4-[(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
{[(3S,4R)-1-[3-(4-fluorophenoxy)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
2-(dimethylamino)-8-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-4-(pyridin-4-yl)pyrimidin-2-amine
N-ethyl-6-fluoro-N-methyl-2-[2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-5-yl]quinoline-4-carboxamide
2-[6-hydroxy-4-(2-methyl-1H-pyrrole-3-carbonyl)-1,4-diazepan-1-yl]-1,3-thiazole-4-carboxamide
N-(3-fluoro-2-methylphenyl)-2-{[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]amino}acetamide
methyl(2-phenylethyl)[(4-{[1-(pyridine-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
{1-[3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)propyl]piperidin-3-yl}methanol
3-(2,5-dioxoimidazolidin-4-yl)-N-[(2-ethoxypyridin-3-yl)methyl]propanamide
3-(3-chloro-1,2-oxazol-5-yl)-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}propan-1-one
2-(dimethylamino)-2-(2-fluorophenyl)-1-{6-oxa-9-azaspiro[4.5]decan-9-yl}ethan-1-one
(2R,6S)-2,6-dimethyl-4-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}morpholine
methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl){[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
{2-[2-(2-ethylphenyl)-1H-imidazol-1-yl]ethyl}dimethylamine
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-2-amine
N,N-dimethyl-2-(1-{[(1-methyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)pyridine-3-carboxamide
8-(5-propylthiophene-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-(2-methylpropyl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-5-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-4-sulfamoylbutanamide
2-(4-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1-(2-methylpropyl)piperazin-2-yl)ethan-1-ol
N-methyl-2-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenoxy)acetamide
4-[(dimethylsulfamoyl)amino]-1-(3-phenylpropyl)pyrrolidin-2-one
2-methyl-N-{3-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenyl}propanamide
1-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-3-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(2,5-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-2,3-dihydro-1-benzofuran-2-carboxamide
(3S,4S)-1-(1-ethyl-1H-pyrazole-3-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-4-(pyridin-2-yl)pyrimidin-2-amine
N,2,6,8-tetramethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]quinoline-4-carboxamide
2-(quinolin-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(1,3-thiazol-2-yl)-decahydro-1,6-naphthyridin-2-one
1-[3-(oxan-4-yl)-1-{[1,2,4]triazolo[4,3-b]pyridazin-6-yl}-1H-1,2,4-triazol-5-yl]ethan-1-ol
N-benzyl-5-(2-chloro-4-methoxyphenoxymethyl)-N-(2-hydroxyethyl)-1,2-oxazole-3-carboxamide
(3S,4R)-3-(dimethylamino)-N-[(4-methoxyphenyl)methyl]-4-propylpyrrolidine-1-carboxamide