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4-[(2-methyl-1,3-oxazol-4-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
3-(3-methoxypyrazin-2-yl)benzoic acid
2-{1-[(2-fluorophenyl)methyl]-4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
4-(3-{2-[(2-methoxyethyl)sulfanyl]-5-(3-methoxyphenyl)pyrimidin-4-yl}piperidine-1-carbonyl)pyridin-1-ium-1-olate
1-(4-carbamoyl-1,3-thiazol-2-yl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-4-(1H-pyrazol-4-yl)butanamide
3-methoxy-1-{2-oxo-2-[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]ethyl}-1,2-dihydropyridin-2-one
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-methyl-1,3-thiazole-4-carboxamide
3-({[(2-methoxyphenyl)methyl](prop-2-en-1-yl)amino}methyl)-N-methylpyridin-2-amine
N-[(1-cyclopentylpiperidin-3-yl)methyl]-1-(1H-imidazol-1-ylmethyl)cyclopropane-1-carboxamide
7-(cyclopropylmethyl)-6-(2-fluoro-4-methoxyphenyl)-2-(pyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]-2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]acetamide
[(2S)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]methanol
1-(2-fluorophenyl)-2-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
3-butyl-4-ethyl-1-{2-oxo-2-[2-(trifluoromethyl)pyrrolidin-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(1-{[4-(2-fluorophenyl)phenyl]methyl}piperidin-4-yl)methyl]acetamide
ethyl 4-({3-[2-hydroxy-3-(morpholin-4-yl)propoxy]phenyl}methyl)piperazine-1-carboxylate
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
(3R,4R)-1-{2-amino-6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-4-cyclobutyl-3-methylpiperidin-4-ol
methyl[(2E)-3-phenylprop-2-en-1-yl][1-(pyrimidin-4-yl)ethyl]amine
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-7-{[(4-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-methyl-4-[3-(2-methylpiperidine-1-carbonyl)phenyl]butan-2-ol
3-{[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-4-propyl-4H-1,2,4-triazole
1-(5-phenyl-1,2,4-oxadiazol-3-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-(1H-pyrazol-1-ylmethyl)cyclopropane-1-carboxamide
9-hydroxy-3-{4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
1-(3-chloro-2-fluorophenyl)-3-(2-methylpropyl)-5-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
3-ethyl-N-[2-(1H-imidazol-4-yl)ethyl]-5-methyl-1,2-oxazole-4-carboxamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
N-[2-(propan-2-yl)phenyl]-N'-[2-(pyridin-3-yloxy)propyl]butanediamide
2-({[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
5-(2-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-oxoethyl)-1,3-dimethylimidazolidine-2,4-dione
2-(3-methoxyphenyl)-1-(1H-1,2,4-triazole-5-carbonyl)piperidine
methyl 5-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propanoyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
(2S,4S)-4-amino-N-methyl-1-[2-(4-methylphenoxymethyl)furan-3-carbonyl]pyrrolidine-2-carboxamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}piperidin-2-one
5-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-{2-[1-(2,3-dihydro-1-benzothiophene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-methyl-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(2-methylpropanoyl)pyrrolidine-2-carboxamide
4-methyl-5-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidine
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-(piperidin-3-yl)benzamide
N-[(6-methylquinolin-5-yl)methyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
(3aS,6aR)-5-(4,6-dimethoxypyrimidin-2-yl)-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[4-(ethylsulfanyl)phenyl]-2-[4-(pyrazin-2-yl)piperazin-1-yl]acetic acid