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N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-[(4S)-2,5-dioxoimidazolidin-4-yl]propanamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][1-(thiophen-2-yl)propan-2-yl]amine
2-[(adamantan-1-ylmethyl)[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]amino]ethan-1-ol
2-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]benzonitrile
N-[2-(dimethylamino)ethyl]-3-{[1-(1-ethylpiperidin-3-yl)piperidin-4-yl]oxy}-N-methylbenzamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(1,3-thiazol-4-ylmethyl)piperidine-4-carboxamide
1-{[3-(propan-2-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-3-ol
2-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-1-yl}propanoic acid
N-(2,4-dimethylphenyl)-2-({[5-(pyridin-2-yl)thiophen-2-yl]methyl}amino)acetamide
N-[4-({7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}methyl)phenyl]acetamide
N-[(1-ethylpiperidin-3-yl)methyl]-3-(2-hydroxyphenyl)propanamide
1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-phenylethyl)piperidine
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[4-methyl-3-(4-methylbenzamido)phenyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
(3S,4R)-1-{[4-(2-aminoethyl)phenyl]methyl}-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
N-[1-(thian-4-yl)piperidin-4-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[(5-{1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazol-4-yl}thiophen-2-yl)methyl]piperidine
1-(pyridin-4-ylmethyl)-4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]-1,4-diazepane
N-(1-hydroxy-2-methylpropan-2-yl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
6-methyl-2-{[({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amino]methyl}quinolin-4-ol
5-{[2-(2-carboxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}furan-2-carboxylic acid
2-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-dimethylacetamide
2-methyl-5-[1-(2-phenylethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-3,4-dihydropyrimidin-4-one
2-[(3-methoxyphenyl)methyl]-8-(5-methyl-1,3-oxazole-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(pyridin-3-yl)ethan-1-one
(4aR,8aR)-4-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-octahydro-2H-1,4-benzoxazine
[3-(3-methoxypropyl)-1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl]methanol
2-methyl-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-[(4-fluoro-3-methylphenyl)methyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-1,4-diazepane
2-(2-phenyl-1,3-thiazol-4-yl)-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}acetamide
7-[(3-phenylphenyl)methyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
methyl 6-(4-methylpentanoyl)-2-[(3-phenylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-cycloheptyl-4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine
N-(3,4-difluorophenyl)-5-[4-hydroxy-1-(thiophen-2-ylmethyl)piperidin-4-yl]-1-benzofuran-2-carboxamide
3-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
3-hexyl-8-(3-methyl-1H-pyrazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{1-[(6-methylpyridin-2-yl)methyl]-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
2,6-dimethyl-4-{[(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)amino]methyl}phenyl acetate
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-2-(2,3-dihydro-1H-inden-1-yl)acetamide
3-[2-(2-methyl-1H-1,3-benzodiazol-1-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{2-[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)amino]ethyl}-1,3-oxazolidin-2-one
1-[2-(dimethylamino)ethyl]-4-[3-(pyridin-2-yl)azetidine-1-carbonyl]pyrrolidin-2-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
N-[2-(furan-2-yl)ethyl]-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
4-(1-propylpiperidin-4-yl)thiomorpholine
3-(2H-1,3-benzodioxol-5-yl)-1-(1,4-oxazepan-4-yl)-3-phenylpropan-1-one
1-{2-[3-(2-methoxyphenoxy)azetidin-1-yl]pyrimidin-4-yl}piperidin-3-ol
(3aR,6aR)-2-methanesulfonyl-5-[(2-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-methylpyrrolidine-2-carboxamide