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2-(2,5-dioxoimidazolidin-4-yl)-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}acetamide
2-{1-[(4-ethylphenyl)methyl]-5-(morpholin-2-ylmethyl)-1H-1,2,4-triazol-3-yl}acetamide
N-(2-phenylethyl)-3-{[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-acetyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidine-4-carboxamide
3-(3-hydroxyphenyl)-3-(4-hydroxyphenyl)-1-[4-(pyrrolidin-1-yl)piperidin-1-yl]propan-1-one
4-{1-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]azetidin-3-yl}pyridine
5-fluoro-2-[1-(1H-indole-6-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
1-[5-({[(5-fluoro-2-methylphenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
2-ethyl-4-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)pyrimidine
5-(2,6-difluorophenoxymethyl)-N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,2-oxazole-3-carboxamide
6-{4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-2-carbonitrile
2-oxo-1-phenyl-N-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]pyrrolidine-3-carboxamide
(4aS,7aR)-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(ethyl)[2-(pyrrolidin-1-yl)ethyl]amine
5-{1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
4-(2-{4-[1-(4-fluorophenyl)cyclopropanecarbonyl]piperazin-1-yl}ethyl)morpholine
2-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-4-amine
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
1-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-ol
2-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-N,N-bis(propan-2-yl)benzamide
1-[5-({[2-(3-chlorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
6-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-7-methylpyrazolo[1,5-a]pyrimidine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-3-(pyridin-4-yl)propan-1-one
1-cyclopropanecarbonyl-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]piperidine-4-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide
4-[1-(4-methoxyphenyl)-5-(2-methyloxolan-2-yl)-1H-1,2,4-triazol-3-yl]pyridine
2-methyl-6-[2-(thiophen-2-yl)azetidine-1-carbonyl]-2,3-dihydropyridazin-3-one
6-[4-(2H-1,3-benzodioxol-5-ylmethyl)-3-oxopiperazin-1-yl]-N,N-dimethylpyridine-3-carboxamide
N-ethyl-2-{4-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]phenyl}acetamide
8-methoxy-2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}quinoline
2-(4,5-dimethyl-1H-imidazol-1-yl)-1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]ethan-1-one
1-cyclohexyl-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N6-cyclopropyl-N5-methyl-N5-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2,5-dimethyl-6-[2-(4-methylpentyl)morpholine-4-carbonyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[(4-methoxyphenyl)methyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
2-methyl-4-({3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)-1,3-thiazole
N-[1-(cyclohex-1-en-1-yl)ethyl]-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
5-(propan-2-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1,2-oxazole-3-carboxamide
2-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}benzonitrile
(2S)-2-amino-3-(4-hydroxyphenyl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]propanamide
4-(1-butyl-1H-imidazol-2-yl)-1-(2-fluorobenzenesulfonyl)piperidine
1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]spiro[azepane-4,2'-chromene]
1-ethyl-6-oxo-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}piperidine-3-carboxamide
4-(6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridazin-3-yl)thiomorpholine
ethyl 2-(1-{4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxyphenyl}-N-methylformamido)acetate
3,5-dimethyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1H-indole-2-carboxamide
1-(cyclopropylmethyl)-3-hydroxy-3-{[4-(6-methylpyridin-2-yl)piperazin-1-yl]methyl}piperidin-2-one
N-[(2,4-dichlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide