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N-(1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
methyl (4aS,7aR)-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
2-(dimethylamino)-2-(3-methylphenyl)-N,N-dipropylacetamide
methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})[4-(morpholin-4-yl)butyl]amine
3-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1-methylpiperidin-4-yl)pyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
[(2,3-difluoro-6-methoxyphenyl)methyl](methyl)[2-(methylamino)ethyl]amine
[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl){[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
3-[(2R,3R,6R)-5-[(3,4-difluorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
5-({4-[6-(piperidin-1-yl)pyrimidin-4-yl]piperazin-1-yl}methyl)pyrimidin-2-amine
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
2-[methyl(2-phenylethyl)amino]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
2-amino-N-[(1R,3R)-3-aminocyclopentyl]-4-methyl-1,3-benzothiazole-6-carboxamide
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-(2-methylpropyl)morpholine
N-(1,3-benzoxazol-2-ylmethyl)-4-[(diethylamino)methyl]-5-ethyl-N-methylfuran-2-carboxamide
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-ol
4-ethyl-1-methyl-3-{1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-phenyl-N-{[8-(pyridin-4-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}butanamide
6-cyclopentyl-N-[3-(1H-imidazol-1-yl)butyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(1-phenylcyclopropanecarbonyl)pyrrolidin-3-yl]methanol
N-[1-(methoxymethyl)cyclopentyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
5-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
1-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-N-(4-fluorophenyl)piperidin-3-amine
2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-N-[2-(4-sulfamoylphenyl)ethyl]-1,4-dihydropyridine-3-carboxamide
(3aS,6aR)-5-(ethanesulfonyl)-3-[3-(4-fluorophenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-(pyridin-2-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]propanamide
4-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carbonyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N-cyclopropyl-3-(2-hydroxyphenyl)-N-[(3-hydroxyphenyl)methyl]-1H-pyrazole-5-carboxamide
1-benzyl-5-{[2-(diethylamino)ethyl](ethyl)amino}azepan-2-one
(2S,4R)-N-ethyl-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[2-(methylsulfanyl)acetamido]pyrrolidine-2-carboxamide
N-(2-methoxyethyl)-2-methyl-N-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
5-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
ethyl 2-cyclohexyl-2-(3-methyl-1H-1,2,4-triazol-5-yl)acetate
2,3-difluoro-6-methoxy-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
6-fluoro-3-[2-(morpholin-4-yl)ethyl]-3,4-dihydroquinazolin-4-one
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-(1-oxo-2,3-dihydro-1H-inden-5-yl)urea
4-(3,4-dihydro-2H-1,5-benzodioxepine-7-sulfonyl)piperazine-2-carboxylic acid
2-amino-6-cyclobutyl-4-(3,4,5-trimethoxyphenyl)pyridine-3-carbonitrile
2-({[2-fluoro-5-(trifluoromethyl)phenyl]methyl}amino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-5-methylpiperidin-2-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-hydroxy-N-methyl-4-(methylsulfanyl)butanamide
[1-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)pyrrolidin-3-yl]methanamine
3-[(2R,3R,6R)-5-[(1-methyl-1H-imidazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
3-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazine
2-(1H-indazol-1-yl)-1-{2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
3-(furan-2-yl)-5-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide