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2-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]acetic acid
N-{2-[({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]ethyl}pyridine-4-carboxamide
3-[(2-fluorophenyl)methoxy]-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)azetidine
[1-(4-fluorophenyl)propyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
2-(1-ethyl-1H-pyrazol-4-yl)-8-methyl-4-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl}quinoline
3-[(2,5-dimethoxyphenyl)methyl]-6,7-dimethoxy-3,4-dihydroquinazolin-4-one
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(2-ethoxyethyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
5-[({[4-(dimethylamino)oxan-4-yl]methyl}carbamoyl)amino]-2-methoxybenzamide
(5S,9aS,9bS)-5-[2-(furan-2-yl)phenyl]-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-cyclohexyl-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[2-(2-ethoxyphenoxy)ethyl]-N-methyl-2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
N-[(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]-2-(phenylsulfanyl)acetamide
methyl 2-{[2-(2-ethoxy-2-oxoethyl)piperidin-1-yl]sulfonyl}benzoate
N-[(4-methoxyphenyl)methyl]-N-(3-methoxypropyl)-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
ethyl 4-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
(2S,4S)-4-amino-1-(3-cyclopentaneamidobenzoyl)-N-methylpyrrolidine-2-carboxamide
(1S,5R)-3-[(5-ethylpyridin-2-yl)methyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
3-[2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]-1,3-oxazolidin-2-one
N-[(4-methoxypyridin-2-yl)methyl]-2,5,6-trimethylpyrimidin-4-amine
5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-N-ethylpyrimidin-2-amine
3-[2-oxo-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]propanoic acid
2-{[(5-chlorothiophen-2-yl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-2-(morpholin-3-yl)acetamide
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-N-[3-(methylsulfanyl)phenyl]piperidine-1-carboxamide
(1S,3R)-3-amino-N-[2-(5-methylfuran-2-yl)ethyl]cyclopentane-1-carboxamide
4-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-amine
2-ethyl-N-({1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}methyl)benzamide
6-(azepan-1-yl)-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-{2-oxo-2-[3-(4-phenoxybenzoyl)piperidin-1-yl]ethyl}-1,3-oxazolidin-2-one
9-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
6-(2-chlorophenyl)-2-(4-{[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
4-{5-[(4-methyl-1H-imidazol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-(3-methylphenyl)-1H-pyrazole
1-ethyl-2,5-dimethyl-N-(1-pentanoylazepan-3-yl)-1H-pyrrole-3-carboxamide
methyl (2R,4S)-4-hydroxy-1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-2-carboxylate
1,3-dimethyl-5-[({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
2,3-dimethyl-7-[3-(pyridin-3-ylmethyl)-1,2,4-oxadiazol-5-yl]-1H-indole
(1-{[methyl({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl})amino]methyl}cyclopropyl)methanol
(1S,4S)-2-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-2-azabicyclo[2.2.1]heptane
2-(1-ethylpiperidin-4-yl)-1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]ethan-1-one
7,8-dimethyl-3-[1-(6-methylpyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
6-{[(5-methyl-1H-imidazol-4-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-(1-cycloheptylpiperidin-3-yl)pyrazine-2-carboxamide
N-(pentan-2-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
N-(2-methoxyethyl)-3-(piperidin-3-yl)-N-(pyridin-4-ylmethyl)benzamide
8-[(2-hydroxy-8-methylquinolin-3-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
2-(methylsulfanyl)-5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyrimidine
2-({[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]amino}methyl)-3,4-dihydroquinazolin-4-one
(1R,9aR)-1-{[(furan-2-ylmethyl)(prop-2-yn-1-yl)amino]methyl}-octahydro-1H-quinolizin-1-ol
2-methyl-4-({methyl[(5-propyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenol