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3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}benzene-1-sulfonamide
2-[2,5-dioxo-4-(piperidin-4-yl)-4-propylimidazolidin-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
5-[1-(4-fluorophenyl)-1H-1,2,4-triazol-5-yl]-N-methylpyrimidin-2-amine
2-(5-methoxy-4-oxo-3,4-dihydroquinazolin-3-yl)-4-methylpentanamide
5-[4-(2-ethoxyphenyl)piperazin-1-yl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N,1,3-trimethyl-N-[(1-methylpyrrolidin-2-yl)methyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(2,2-diphenylacetyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-1H-imidazole-2-carboxamide
2-benzyl-4-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[2-(dimethylamino)ethyl]-N-[(6-methylpyridin-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
4-{2-[3-(morpholine-4-carbonyl)piperidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
(3S,9aR)-3-(cyclohexylmethyl)-8-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3S,9aR)-8-benzoyl-3-[(2S)-butan-2-yl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
2-methoxy-1-{4-[4-(pyridin-4-yl)piperazine-1-carbonyl]piperidin-1-yl}ethan-1-one
(3aS,6aS)-2-(cyclopropylmethyl)-5-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-methyl-5-{2-[4-(2-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(carbamoylmethyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]piperidine-4-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazole
N-[(3R,4S)-1-(1-acetylpiperidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]pyridazine-3-carboxamide
8-fluoro-2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}quinoline
5-{3-[2-(ethylsulfanyl)pyrimidin-5-yl]-3-(morpholin-4-yl)prop-1-yn-1-yl}pyridin-2-amine
N-(2-methoxyethyl)-6,6-dimethyl-5-oxo-N-(pyridin-2-ylmethyl)thiomorpholine-3-carboxamide
4-methyl-2-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}pyrimidine
4-(piperidin-1-ylmethyl)-N-[2-(pyrazin-2-yl)ethyl]benzamide
2-amino-6-(4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)pyrimidin-4-ol
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(1,3-thiazol-2-yl)piperidine
N-cyclopropyl-1-[1-(5-methylthiophene-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
ethyl 2-{8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl}-1,3-oxazole-4-carboxylate
[3-(3-methylbut-2-en-1-yl)-1-(pyrimidin-2-ylmethyl)piperidin-3-yl]methanol
[(4-fluoro-3-methoxyphenyl)methyl](methyl)[(3-methyl-1H-pyrazol-4-yl)methyl]amine
2-methyl-5-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]pyrimidin-4-ol
2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-cyclopentyl-1,4-diazepane
4-{5-[(dimethylamino)methyl]furan-2-carbonyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
5-(5-chlorothiophen-2-yl)-3-methyl-1H-1,2,4-triazole
4-(4-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]amino}piperidin-1-yl)-6-methylpyrimidin-2-amine
1-methyl-N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-butyl-N,5-diethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
5-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-(4-{[(adamantan-1-ylmethyl)(methyl)amino]methyl}phenoxy)-3-(dimethylamino)propan-2-ol
N-[(1-ethyl-1H-indazol-3-yl)methyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
4-methyl-N-(2-methylpropyl)-2-(pyridin-3-yl)-N-(thiophen-3-ylmethyl)pyrimidine-5-carboxamide
N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
1-(3-chloro-2-propoxyphenyl)-3-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}urea
2-{1-cyclopentyl-4-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-{2-[1-(3,4-dimethoxybenzenesulfonyl)piperidin-2-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-(2-ethylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4R)-1-[(5-ethylfuran-2-yl)methyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid