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1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
1-(2-methoxyacetyl)-N-{[1-(pyridin-2-yl)piperidin-3-yl]methyl}piperidine-4-carboxamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,2-dihydroquinoxalin-2-one
N-{4-[2-amino-3-cyano-6-(trimethyl-1H-pyrazol-4-yl)pyridin-4-yl]phenyl}acetamide
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-(3-methylbenzoyl)piperidine
2-(4-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}morpholin-3-yl)-1-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
N-ethyl-5-(3-fluorophenoxymethyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazole-3-carboxamide
[(2,4-difluorophenyl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
3-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclohexyl-5-(3-methyl-1H-pyrazol-1-yl)furan-2-carboxamide
4-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-6-(piperidin-4-yl)pyrimidin-4-amine
4-({1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-yl}methyl)benzoic acid
4-[(2-ethoxyphenyl)methyl]-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-methanesulfonyl-4-(piperidin-3-yl)-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrimidine
2-(2-{[1-(1,3-benzothiazol-2-yl)piperidin-4-yl]amino}ethyl)-6-methyl-3,4-dihydropyrimidin-4-one
4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}-N-(2-phenylethyl)piperidine-1-carboxamide
1-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
N-benzyl-N-(2-hydroxyethyl)-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
1-cyclopentyl-N3-ethyl-N5-[(2-methoxynaphthalen-1-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(furan-2-ylmethyl)-N-(1-hydroxy-2-methylpropan-2-yl)-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-[1'-(3-fluoropyridin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
(2S)-1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(methylamino)propan-1-one
5-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
N-butyl-2-[N-methyl-1-(3,5,7-trimethyl-1H-indol-2-yl)formamido]acetamide
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(thiophen-3-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
4-(2-propyl-1H-imidazol-1-yl)thiophene-2-carboxamide
1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-4-(hydroxymethyl)azepan-4-ol
6-(2-chlorophenyl)-N-(1,3-dihydroxypropan-2-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[3-(1H-imidazol-1-yl)propyl]-1,2-dihydroquinoxalin-2-one
N-(2-hydroxyethyl)-5-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-ethyl-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aS,6aS)-2-(1H-indol-5-ylmethyl)-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(4-{[(6-methoxypyrimidin-4-yl)amino]methyl}piperidin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
ethyl({[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}){[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
methyl(quinolin-6-ylmethyl)[(4-{[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(2S)-2-(methoxymethyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-1-carboxamide
ethyl 1-{[2-(furan-2-yl)phenyl]methyl}-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
({4-ethyl-5-[1-(2-phenylethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-[3-(dimethylcarbamoyl)-4-hydroxyphenyl]-5-oxopyrrolidine-3-carboxylic acid
2-(2-{3-[(1-methylpiperidin-4-yl)methyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}ethyl)pyrazine
N-{4-[(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)methyl]phenyl}acetamide
6-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]pyridine-2-carbonitrile
N-[2-(propan-2-yloxy)ethyl]-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
8-(1-methyl-1H-imidazole-5-carbonyl)-2-(pyridin-2-yl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-[2-({1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}amino)ethyl]-1,3-oxazinan-2-one
2-[5-(2-fluoro-4-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]-N-methylethane-1-sulfonamide
5-acetyl-6-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine