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N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-8-fluoro-4-oxo-1,4-dihydroquinoline-2-carboxamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(2-oxopiperidin-1-yl)acetamide
2-{methyl[3-(1H-pyrazol-1-yl)propyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
ethyl 4-{[4-(1H-pyrrole-2-carbonyl)piperazine-1-carbonyl]amino}benzoate
4-(5-phenyl-1,2,4-oxadiazol-3-yl)-1,4-oxazepan-6-ol
3-methyl-7-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(3-hydroxyazetidin-1-yl)pyridine-3-carboxamide
2-{1-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}quinoline
(3aS,6aS)-2-(ethanesulfonyl)-5-[(2-methyl-1,3-oxazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(ethanesulfonyl)acetamide
6-[5-(2-ethylpyrimidin-4-yl)-4-phenyl-1H-imidazol-1-yl]-2-methylheptan-2-ol
(2E)-1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-3-phenylprop-2-en-1-one
1-(3-chloro-4-fluorophenyl)-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazine
(1S,5R)-6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
[1-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(4-fluorophenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[2-(4,6-dimethylpyrimidin-2-yl)ethyl]amine
2-(4-{[3-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
4-(4-ethyl-1H-pyrazol-5-yl)-1-[3-(4-ethylphenyl)-1H-pyrazole-5-carbonyl]piperidine
5-{1-[(2,6-difluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(1,4-dioxan-2-ylmethyl)-1-benzofuran-2-carboxamide
3-({[2-(dimethylamino)ethyl][(5-methylthiophen-2-yl)methyl]amino}methyl)piperidin-3-ol
14-[4-(pyrimidin-2-yloxy)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
(3R,4R)-4-(azepan-1-yl)-1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-ol
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
1-({[1-(furan-2-ylmethyl)piperidin-4-yl]formamido}methyl)cyclopentane-1-carboxylic acid
N-methyl-2-(5-oxo-1-phenyl-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)-N-(thian-4-yl)acetamide
1-(4-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}phenyl)-1H-1,2,4-triazole
2-[1-(2,5-dimethylfuran-3-carbonyl)pyrrolidin-2-yl]pyridine
2-{4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
1-{2,7-diazaspiro[4.5]decan-2-yl}-2-[(4-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
4-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1-phenylpiperazin-2-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(5-ethyl-1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(1s,5s)-3,7-dimethyl-10-(4-methylpyrimidin-2-yl)-3,7,10-triazatricyclo[3.3.3.01,5]undecane
N-(3,3-diphenylpropyl)-3-(2-ethyl-5-oxopyrrolidin-2-yl)propanamide
1-methyl-5-[methyl(2-methylpropyl)amino]-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[4-(2-benzyl-1,3-thiazole-4-carbonyl)morpholin-3-yl]acetic acid
4-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}-2-ethoxyphenol
2-(3,4-dimethylphenyl)-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]acetic acid
N-[3-(2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]-5-phenylpentan-1-one
3-{2-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
N-{[1-(2-chloropyridine-4-carbonyl)piperidin-3-yl]methyl}-3,5-dimethoxybenzamide
1-(2-methoxyacetyl)-N-{2-[methyl(phenyl)amino]ethyl}piperidine-3-carboxamide
N-(2-hydroxyethyl)-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-benzyl-3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]propanamide
1-benzyl-3-(2-methoxyethyl)-8-(1-methoxypropan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(5-fluoro-2-methoxyphenyl)-2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}acetic acid
N-[(2-methoxynaphthalen-1-yl)methyl]-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
1-(1-benzylpiperidin-3-yl)-4-(2-methylphenyl)piperazine
(1S,5R)-6-benzyl-3-(5-methylpyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one