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1-{5-methoxy-2-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
2-methyl-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
(3S,5R)-1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-1H-pyrazole-4-carboxamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[5-(2-methyl-4-phenylpyridin-3-yl)-2H-1,2,3,4-tetrazol-2-yl]acetamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
2-(4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-5-methyl-2-oxopiperazin-1-yl)benzonitrile
4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-2-amine
N-[(3R,4S)-1-(2-methyl-6-propylpyrimidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N,N-dimethyl-4-[(1E)-3-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]prop-1-en-1-yl]aniline
N,N-dimethyl-4-[3-(1,2-oxazinane-2-carbonyl)phenoxy]piperidine-1-sulfonamide
1-cyclopentyl-4-(1-cyclopropyl-6-oxopiperidine-3-carbonyl)piperazin-2-one
2-(dimethyl-1,2-oxazol-4-yl)-1-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
2-{4-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl}acetic acid
6-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]quinoxaline
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)ethyl]acetamide
2-(2-chlorophenyl)-N,3-dimethyl-N-(pyrimidin-4-ylmethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
3-[(3-hydroxyazetidin-1-yl)methyl]-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
N-{4-[(2H-1,3-benzodioxol-5-ylmethyl)carbamoyl]-2-methylphenyl}furan-2-carboxamide
3-(thiomorpholine-4-sulfonyl)-5-(thiophen-3-yl)benzoic acid
(2,1,3-benzoxadiazol-5-ylmethyl)[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl]amine
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
N4-[(2-chloro-4-fluorophenyl)methyl]-6-methylpyrimidine-2,4-diamine
N-methyl-6-[(oxan-2-ylmethyl)amino]-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
{1-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
5-[3-hydroxy-3-(2-methylphenyl)pyrrolidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidin-4-ol
3-[(2-hydroxyadamantan-2-yl)methyl]-1-[4-(methylsulfanyl)phenyl]urea
N4-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
2-[4-(4-chloro-3-fluorophenyl)-1H-pyrazol-1-yl]ethan-1-ol
N-[(2E)-3-phenylprop-2-en-1-yl]-N-propyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
4-(2-hydroxybutyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2R,6S)-4-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,6-dimethylmorpholine
N-[(5-chloro-2-propoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
4-[(4-methylphenyl)sulfanyl]-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine
1-[2-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethyl]cyclopentan-1-ol
3-methyl-1-{4-[2-(pyridin-2-yl)ethoxy]phenyl}-3-(thian-4-yl)urea
3-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-N-(6-methylpyridazin-3-yl)benzamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[2-(3-methoxyphenyl)piperidin-1-yl]propan-1-one
4-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenol
N-methyl-2-(phenylamino)-N-(quinolin-5-ylmethyl)pyrimidine-5-carboxamide
4-[4-(4-fluoropiperidine-1-carbonyl)phenyl]-2-methylbutan-2-ol
2,3,5,6-tetramethyl-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]benzamide
2-(4-methyl-6-{4-[(pyridin-3-ylmethyl)amino]piperidin-1-yl}pyrimidin-2-yl)phenol
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxylic acid
4-({4-[(3-chlorophenyl)methyl]piperazin-1-yl}methyl)-1,5-dimethyl-1H-pyrrole-2-carbonitrile
(1S,4S)-2-(3-chloro-4-methoxyphenyl)-5-[2-(4-fluorophenyl)acetyl]-2,5-diazabicyclo[2.2.1]heptan-3-one