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2-{[(prop-2-en-1-yl)(pyridin-3-ylmethyl)amino]methyl}pyridine-3-carboxylic acid
3-{1-[(1R,7S)-3-[(3-methoxyphenyl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-6-yl]-N-methylformamido}propanamide
(1R,4S)-2-[2-(1H-pyrazol-4-yl)pyridine-3-carbonyl]-2-azabicyclo[2.2.1]heptane
(2S,4S)-4-amino-1-[4,5-dimethyl-2-(1H-pyrrol-1-yl)thiophene-3-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-{5-[(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)methyl]-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl}acetamide
9-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)methyl]pyrrolidin-3-ol
4-{1-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1H-imidazol-2-yl}benzoic acid
N1-{3-[(2-methoxyethyl)carbamoyl]-2-methylphenyl}piperidine-1,4-dicarboxamide
5-[2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1R,5R)-3-cyclobutanecarbonyl-6-[(1-propyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-(3-chlorophenyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]-3-phenylpropanamide
6-methoxy-3-methyl-N-[2-(pyridin-3-yl)ethyl]-1-benzofuran-2-carboxamide
3-(4-chlorophenyl)-N-[(2-methylpyridin-4-yl)methyl]-3-phenylpropanamide
(2E)-1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-(4-methoxyphenyl)prop-2-en-1-one
ethyl 1-[(3-ethoxy-3-oxopropyl)carbamoyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
2-{[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]amino}-N-(pyrazin-2-yl)acetamide
(4aS,8aR)-1-(3-aminopropyl)-N-[(4-methylphenyl)methyl]-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
4-[(2-fluoro-5-methoxyphenyl)methyl]-5-methyl-1-(2-methylphenyl)piperazin-2-one
2-(2,5-dioxoimidazolidin-1-yl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]cyclopentanecarboxamide
(1R,5R)-6-{[4-(methylsulfanyl)phenyl]methyl}-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-amino-1-[7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]ethan-1-one
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-1,3-benzothiazole-6-carboxamide
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,N-dimethylacetamide
4-({3-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]phenyl}methyl)piperidine
N-(cyclopropylmethyl)-1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidine-3-carboxamide
3-{[(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
2-(pyridin-3-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
2-[(1-ethylpyrrolidin-2-yl)methyl]-4-(4-fluoropiperidine-1-carbonyl)-2,3-dihydro-1H-isoindol-1-one
{7-[5-(1H-1,3-benzodiazol-2-yl)furan-2-yl]-4-fluoro-2,3-dihydro-1-benzofuran-2-yl}methanamine
3-({3-[(2-methoxyphenyl)methyl]-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl}methyl)-1,3-oxazolidin-2-one
4-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-6-methylpyrimidin-2-amine
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
2-[1-(3-phenylpropyl)-4-(pyrazine-2-carbonyl)piperazin-2-yl]ethan-1-ol
ethyl 1-benzyl-5-[(4-methyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[1-(4-methanesulfonylphenyl)propyl]-2-methyl-1,3-thiazole-4-carboxamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1,2-oxazole-3-carboxamide
dimethyl(3-{3-[3-(3-methylpyridin-2-yl)phenyl]-1H-pyrazol-1-yl}propyl)amine
8-[3-(3-hydroxy-3-methylbutyl)benzoyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-{4-[(6,7-dimethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperazin-1-yl}acetamide
N-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-ethylbenzamide
[(2-butyl-1H-imidazol-4-yl)methyl](2-methoxyethyl)(thiophen-2-ylmethyl)amine
(2-methoxy-5-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methanol
3,3-dimethyl-1-[(5-{[3-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]urea
8-oxo-7-(prop-2-en-1-yl)-N-propyl-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[(8-methoxyquinolin-5-yl)methyl]-N,5-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide