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N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-5-propyl-1,3,4-oxadiazole-2-carboxamide
2-({[2-(2-methoxyethoxy)phenyl]carbamoyl}amino)-N,N-dimethyl-2-phenylacetamide
2-[2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(2E)-1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-(pyridin-4-yl)prop-2-en-1-one
8-(furan-3-carbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(oxolane-2-carbonyl)-4-[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperazine
N-[(3R,4S)-1-(2-aminopyrimidin-4-yl)-4-propylpyrrolidin-3-yl]-2-acetamido-2-methylpropanamide
methyl 1-({3-[(pyridin-4-yl)carbamoyl]phenyl}methyl)pyrrolidine-2-carboxylate
1-cyclohexyl-N3-[2-(3-fluorophenyl)ethyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-(1-hydroxybutan-2-yl)-1-(3-methylcinnolin-5-yl)-3-[(5-methylthiophen-2-yl)methyl]urea
2-amino-4-(4-hydroxy-2-methoxyphenyl)-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-4-(1H-pyrazol-3-yl)benzamide
1-phenyl-4-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)piperazine
1-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-yl}-2-(morpholin-4-yl)ethane-1,2-dione
1-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(1-propyl-1H-1,3-benzodiazol-5-yl)urea
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-(3-methylthiophene-2-carbonyl)piperidine
3-(3,3-diphenylpiperidin-1-yl)-N-methylpropanamide
4-{4-[2-(2-ethylphenoxy)ethyl]-2-oxopiperazin-1-yl}benzonitrile
N-[(5-methoxy-1H-indol-2-yl)methyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-3-(pyridin-3-yl)propan-1-one
3-({[2-(2,5-dimethylphenyl)ethyl]amino}methyl)-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
3-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]-6-(propan-2-yl)pyridazine
7-(2-fluoro-5-methoxyphenyl)-1,2,3,4-tetrahydroisoquinoline
4-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-2-(propan-2-yl)pyrimidine
2-cyclopentyl-1-[1-methyl-4-(3,3,3-trifluoropropyl)-1,4,9-triazaspiro[5.5]undecan-9-yl]ethan-1-one
5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-1H-indole
ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
1-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
4-{[(1,2-dimethyl-1H-imidazol-5-yl)methyl]amino}-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
ethyl 4-({1-[3-(2-methoxybenzamido)phenyl]piperidin-4-yl}amino)piperidine-1-carboxylate
(3S,4R)-1-[1-(dimethylcarbamoyl)piperidine-4-carbonyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
1-methyl-3-(propan-2-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-ol
N-(benzylsulfamoyl)-N-[(2-chlorophenyl)methyl]cyclopropanamine
4-(2,6-dimethylpyridin-3-yl)-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-2-amine
9-methoxy-7-[4-(methylsulfanyl)phenyl]-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[4-(furan-3-carbonyl)-1,4-diazepane-1-carbonyl]-3,5-dimethyl-1H-indole
2-(3-phenylpropyl)-N-[3-(propan-2-yloxy)propyl]-1,3-benzoxazole-5-carboxamide
2-(4-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}phenyl)ethan-1-amine
2-[({5-[1-(1H-imidazole-2-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)furan-3-carboxamide
2-methoxy-6-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)phenol
(4aS,7aR)-1-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanoyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,4-dimethoxy-N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)benzamide
2-[1-(2-methylpropyl)-4-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl]ethan-1-ol
1-(2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenyl)ethan-1-one
N-(1,3-thiazol-2-yl)-3-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propanamide
methyl 3-[(cyclobutylformamido)methyl]-5-[3-(trifluoromethyl)benzamido]benzoate
1-[1-(4-cyanopyridin-2-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide