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2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)butanamide
2-{2-[1-(3-chloro-2-fluorophenyl)-1H-imidazol-2-yl]phenoxy}ethan-1-ol
5-methoxy-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-4-oxo-4H-pyran-2-carboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(5-phenyl-1,2-oxazole-4-carbonyl)piperidine
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-1-phenylcyclopropane-1-carboxamide
4-(2-{1-cyclohexyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-2-methylpropyl)morpholine
2-{2-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-1H-pyrrol-1-yl}pyrimidine
(3S)-1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-N,N-dimethylpyrrolidin-3-amine
2-methyl-6-(piperidin-4-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]pyrimidin-4-amine
N-[(2-fluorophenyl)methyl]-3-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}propanamide
1-[cyclohexyl(methyl)amino]-3-(2-{[(2-phenoxyethyl)amino]methyl}phenoxy)propan-2-ol
(3R,4R)-4-{[6-methyl-2-(methylsulfanyl)pyrimidin-4-yl]amino}piperidin-3-ol
7-(pyridin-3-yl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yloxy)ethyl]acetamide
[(3R,4R)-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(1H-indol-3-yl)acetamide
(3S,4S)-4-propyl-1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}pyrrolidine-3-carboxylic acid
N-{3-[cyclopentyl(methyl)amino]propyl}-4-ethyl-5-methylpyrimidin-2-amine
3-[(3R,4S)-1-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-(1,5-dimethyl-1H-indazole-3-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
2-({3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-5-methoxyphenol
(1S,5R)-3-benzyl-6-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
N-({1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl}methyl)-2,1-benzoxazole-3-carboxamide
4-methyl-2-oxo-5-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridine-3-carbonitrile
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(1H-pyrazole-3-carbonyl)-1,4-diazepan-5-one
8-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[(4-methanesulfonylmorpholin-2-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(5S)-5-[({[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}(pyridin-3-ylmethyl)amino)methyl]pyrrolidin-2-one
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[1-(2-methylpropyl)-4-(pyridin-2-ylmethyl)piperazin-2-yl]ethan-1-ol
1-[2-(1H-imidazol-4-yl)ethyl]-3-[5-(4-methylphenoxymethyl)-1,3,4-thiadiazol-2-yl]urea
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine
8-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(1-methylpiperidin-4-yl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
N-methyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(morpholin-4-yl)ethyl]acetamide
4-[1-butyl-5-(oxolan-3-ylmethyl)-1H-1,2,4-triazol-3-yl]pyridine
N-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
6-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
4-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
8-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
7-fluoro-2-oxo-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-1,3-benzothiazole
(4aS,7aR)-1-(4-methylpentanoyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[4-(2-methylphenyl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
2-(cyclopent-2-en-1-yl)-N-{[1-(hydroxymethyl)cyclopentyl]methyl}acetamide
3-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}-N-(1-methyl-1H-1,2,4-triazol-3-yl)benzamide
N-(2-methoxyethyl)-2-(methylamino)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyridine-4-carboxamide
1-[(4-chlorophenyl)methyl]-6-oxo-N-{2-[(pyridin-3-yl)amino]ethyl}piperidine-3-carboxamide
N-{1-[1-(2-methylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
N-[(3S,4R)-1-[(8-methoxy-2H-chromen-3-yl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide