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3-({1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}carbamoyl)benzoic acid
6-({8-[2-(dimethylamino)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
8-{3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]propanoyl}-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(4aS,8aR)-1-(2-aminoethyl)-6-[3-(pyridin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
1-(cyclohexylmethyl)-6-oxo-N-{2-[(pyridin-3-yl)amino]ethyl}piperidine-3-carboxamide
2-(3-hydroxypropyl)-9-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2,9-diazaspiro[5.5]undecan-3-one
8-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-1-oxa-8-azaspiro[4.5]decane
7-propyl-2-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-cyclobutyl-N-(3-phenylpropyl)-1,3,4-oxadiazol-2-amine
(3aS,6aS)-2-cyclopentyl-5-(4-ethenylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-3-yl}-4-methyl-1,3-thiazol-2-amine
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]propan-1-one
2-methyl-5-{4-[3-(2-methylphenoxy)azetidine-1-carbonyl]phenyl}-2H-1,2,3,4-tetrazole
5-(ethanesulfonyl)-2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(3S,4S)-3-hydroxy-4-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]-1λ6-thiolane-1,1-dione
4-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
N-[(3S)-1-benzylpyrrolidin-3-yl]-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
(1R,5R)-6-(cyclopropylmethyl)-3-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-methoxypyrazine
5-chloro-N-[3-methoxy-4-(3-methylbutanamido)phenyl]pyridine-2-carboxamide
(4aS,8aR)-6-[5-(methoxymethyl)thiophene-2-carbonyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
2-{4-[6-(cyclopentylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-1-yl}-N,N-dimethylacetamide
N-(4-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}phenyl)acetamide
2-[(2S)-2-aminohexanoyl]-N-cyclobutyl-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-cyclopropyl-5-oxo-N-[2-(2-phenoxyphenyl)ethyl]pyrrolidine-3-carboxamide
3-{1-[1-(3,4-dimethylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
4-{3-[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]propoxy}benzamide
1-[2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-4-phenylpiperazine
3-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-ylmethyl]-N-(5-fluoropyridin-2-yl)benzamide
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-2-methyl-5-(propan-2-yl)furan-3-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]quinoxalin-6-amine
ethyl 1-(2-hydroxyethyl)-5-[(5-methylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-3-ylmethyl)acetamide
3-(2-oxoazepan-1-yl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)propanamide
4-{2-[2,5-dioxo-4-(piperidin-4-yl)-4-propylimidazolidin-1-yl]ethyl}benzonitrile
5-[2-(1H-imidazol-5-yl)-1-(1H-pyrrol-1-yl)ethyl]-3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazole
2-(2-hydroxyethyl)-9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-N,N-diethylpyrrolidin-3-amine
1-[(5-chlorothiophen-2-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
[4-benzyl-1-(8-methoxyquinolin-2-yl)piperidin-4-yl]methanol
1-ethyl-4-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
{[4-(6-ethylpyrimidin-4-yl)-1,4-oxazepan-6-yl]methyl}dimethylamine
(1S,6R)-9-[1-methyl-5-(trifluoromethyl)-1H-pyrazole-3-carbonyl]-3,9-diazabicyclo[4.2.1]nonane
4-chloro-3-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-pyrazol-5-amine
(3aR,6aR)-2-cyclopentanecarbonyl-5-(5-propyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(1-benzyl-1H-imidazol-2-yl)methyl](methyl)[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]amine
4-(1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidine-3-carbonyl)morpholine
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid