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N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(2-ethyl-1H-imidazol-1-yl)acetamide
2-fluoro-N-{3-[4-(2-methylpropyl)piperazin-1-yl]-3-oxopropyl}benzamide
8-(5-phenyl-1,2,4-oxadiazol-3-yl)-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-(methoxymethyl)-N-methylpyrimidin-4-amine
N-[2-(azepan-1-yl)ethyl]-3-chloro-N-ethylpyridine-4-carboxamide
1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
1-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3-benzotriazole
1-(cyclohex-3-ene-1-carbonyl)-4-[(2,6-dimethylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
7,7-dimethyl-2-[2-(pyridin-4-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[4-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]-1-(morpholin-4-yl)ethan-1-one
3-({3-[3-(2-methoxyphenyl)phenyl]-1H-pyrazol-1-yl}methyl)-5-methyl-1,2-oxazole
N-methyl-N-(2-methylpropyl)-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
2-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}-N-(pyrazin-2-yl)acetamide
N-methyl-5-({[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amino}methyl)-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
6-(2-methoxypyridin-3-yl)pyridine-2-carbonitrile
4-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]-1-(propan-2-yl)pyrrolidin-2-one
2-(2-{1-cyclopentyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrrol-1-yl)-1,3-thiazole
2-(4-chloro-2-methoxy-6-{[methyl(1-methylpiperidin-4-yl)amino]methyl}phenoxy)propanoic acid
8-{[4-(trifluoromethoxy)phenyl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
3-ethyl-1-methyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-1H-pyrazole-5-carboxamide
methyl[(1-phenyl-1H-pyrazol-5-yl)methyl][1-(pyridin-2-yl)ethyl]amine
ethyl 1-(pyridin-2-yl)-5-(thiomorpholin-4-ylmethyl)-1H-pyrazole-4-carboxylate
2-(4-chlorophenyl)-4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}morpholine
1-[(3-methylpyridin-2-yl)methyl]-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
4-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-phenylbutan-1-one
5-[3-(thiophen-3-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidin-3-ol
5-(propan-2-yl)-N-(1,3-thiazol-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
5-benzyl-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-{2-[1-(4-methoxyphenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
1-methyl-5-{[1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-yl]amino}piperidin-2-one
5-benzamido-1-cyclopentyl-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-1H-1,3-benzodiazole-7-carboxamide
5-[(3-methoxypyrrolidin-1-yl)methyl]-2-(pyridin-2-yl)pyrimidine
5-methoxy-9-(2-methylquinoline-4-carbonyl)-1-oxa-9-azaspiro[5.5]undecane
(4aR,7aS)-1-methanesulfonyl-4-(1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-fluoro-5-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
N-[(3S,4R)-4-propyl-1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]methanesulfonamide
(1S,5R)-3-(7-fluoro-2-methylquinoline-4-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,5R)-6-methyl-3-[3-(1H-pyrrol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
2-(3,4-dichlorophenyl)-1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}ethan-1-one
4-[6-methyl-2-(methylsulfanyl)pyrimidin-4-yl]-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
[3-benzyl-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl]methanol
N-[3-(morpholin-4-yl)propyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(thiophen-2-yl)propanamide
5-[(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(2-benzyl-1,3-thiazole-4-carbonyl)-4-(pyrimidin-2-yl)-1,4-diazepane
4-{[1-(phenylcarbamoyl)pyrrolidin-3-yl]methyl}benzoic acid
2-(1-ethylpiperidin-4-yl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide