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4-{2-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-2-methylpropyl}morpholine
2-[4-(dimethylamino)phenyl]-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
2-[5-(3-ethyl-1H-indol-2-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
2-methyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[1'-(4-ethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-(pyrimidin-2-yl)piperidin-4-amine
6-[3-(1H-pyrazol-5-yl)piperidin-1-yl]pyridine-3-carbonitrile
1-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
3-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-3-yl]benzoic acid
3-{3-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-3-oxopropyl}-3,4-dihydroquinazolin-4-one
8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(3-{[(4-fluorophenyl)methyl]sulfanyl}propanoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
3-[2-(dimethylamino)ethyl]-5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
3-amino-1-{[5-(2-cyanophenyl)furan-2-yl]methyl}pyrrolidine-3-carboxylic acid
2-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5-chlorophenol
N,2,3-trimethyl-N-[2-(oxan-2-yl)ethyl]quinoxaline-6-carboxamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]piperidine-4-carboxylic acid
3-(3-methoxyphenyl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1H-pyrazole-4-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-{3-[(2-methoxyphenyl)methyl]-5-(oxan-2-yl)-1H-1,2,4-triazol-1-yl}-4-methylpyridine
3-methoxy-1-{2-oxo-2-[3-(propoxymethyl)pyrrolidin-1-yl]ethyl}-1,2-dihydropyridin-2-one
1-(1-benzylpiperidine-2-carbonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
2-(cyclopropylmethyl)-3-oxo-N-[(1R)-1-phenylethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
7-methoxy-3-({[1-(methoxymethyl)cyclopropyl](methyl)amino}methyl)-1,2-dihydroquinolin-2-one
9-methoxy-7-[4-(methylsulfanyl)phenyl]-4-(quinolin-8-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[1-(1H-1,3-benzodiazol-2-ylmethyl)-4-phenylpiperidin-4-yl]ethan-1-one
4-{[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
4-[(2-fluorophenyl)methyl]-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{4-oxo-4-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butyl}acetamide
2-({2-[1-(4-methoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
1-[2-(methylsulfanyl)benzoyl]-4-(2-phenoxyethyl)piperazine
(3S,4S)-4-(4,4-difluoropiperidin-1-yl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)pyrrolidin-3-ol
4-(3-hydroxy-3-methylbutyl)-N-[1-(3-methylphenyl)-5-oxopyrrolidin-3-yl]benzamide
3-methyl-8-[2-(2-oxo-1,2-dihydroquinolin-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5-(3-ethynylbenzoyl)-3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3-(3-methoxyphenoxymethyl)piperidine
3-[(4aR,7aS)-6,6-dioxo-4-(2,2,3,3-tetramethylcyclopropanecarbonyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-({5-[(3-chloro-2,6-difluorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
5-[(4aS,7aR)-4-(2-methoxyacetyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]pyridine-2-carbonitrile
N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]azocane-1-carboxamide
methyl 6-[(3-chlorophenyl)methyl]-2-[methyl(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(furan-2-yl)ethyl]-1H-pyrazole-3-carboxamide
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-(1-methyl-1H-imidazol-2-yl)piperidine
8-(1H-imidazol-2-ylmethyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[4-(thiophen-2-yl)butanoyl]pyrrolidin-3-yl]urea
4-{1-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-propyl-5-{[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidin-2-amine
3-[3-(propan-2-yloxy)benzoyl]-1-(1-propylpiperidin-4-yl)piperidine
5-methoxy-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-methyl-1H-indole-2-carboxamide