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N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(oxolan-2-ylmethyl)amine
5-methyl-3-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,2-oxazole
1-[(5-chlorothiophen-2-yl)methyl]-5-{2-[(2-phenoxyethyl)amino]ethyl}pyrrolidin-2-one
1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-N-(4-fluorophenyl)piperidin-3-amine
methyl 3-acetamido-1-[2-(1H-indol-3-yl)ethyl]-5-[(4-methylpentan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(1-benzylpyrrolidin-3-yl)-3-{1-[3-(pyrazin-2-yl)propanoyl]piperidin-4-yl}propanamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)benzamide
1-(3-phenylpropyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
6-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,3-dihydropyridazin-3-one
3-[(2-chlorophenyl)methyl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-2-[3-(3-methylphenoxy)azetidin-1-yl]pyrimidine
{[5-(4-chlorophenyl)furan-2-yl]methyl}({3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl})amine
6-fluoro-4-[2-(1-methylpiperidin-2-yl)ethyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-({1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-3-ethylurea
4-(cyclopropylmethyl)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-(propan-2-yl)-1,4-diazepan-5-one
5-fluoro-2-(quinolin-3-yl)phenol
2-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-1H-imidazole
8-(8-methoxy-4-methylquinolin-2-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
({3-[(1-cyclohexanecarbonylpiperidin-4-yl)oxy]phenyl}methyl)(methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
1-(2-methylpropyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
2-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-[2-(thiophen-2-yl)ethyl]-1H-imidazole
6-methyl-3-(4-methylpiperidine-1-carbonyl)-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridin-4-one
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(3-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(2-fluorophenyl)methyl]-4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
3-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-[1-(4-methylpyridin-2-yl)propyl]urea
N-methyl-N-[2-(phenylsulfanyl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-(1-methylcyclopropanecarbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-methyl-N-(3-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-3-oxopropyl)methanesulfonamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-cyclopentanecarbonylpiperidine-4-carboxamide
4-(5-chloro-2-fluorobenzoyl)-1-(4-methylphenyl)piperazin-2-one
2-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonane-7-carbonyl]benzonitrile
2-ethyl-N-(furan-2-ylmethyl)-N-(2-hydroxyethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[2-(pyridin-3-yloxy)phenyl]-1H-pyrazole-4-carboxamide
N-{1-[1-(2-oxo-2H-chromene-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
1-[(2-chlorophenyl)methyl]-4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
ethyl 1-[(5-acetylthiophen-3-yl)methyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
2-methoxy-4-[(1E)-3-{4-[5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}prop-1-en-1-yl]phenol
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-3-(2-fluorophenyl)propan-1-one
(3S,4R)-1-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
(3S,4R)-1-(5-methoxypyrimidin-2-yl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
4-benzyl-3-ethyl-1-(5-ethyl-1,3-oxazole-4-carbonyl)-1,4-diazepan-5-one
(3S,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
2,3-difluoro-5-(2-propyl-1H-imidazol-1-yl)phenol
2-methyl-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
N-[(3S,4R)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
3-[1-(2-chloro-4-fluorobenzoyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
1-ethyl-4-{[methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}-1H-pyrrole-2-carbonitrile