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ethyl 3-[(2-methylphenyl)methyl]-1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidine-3-carboxylate
(4aS,7aR)-1-(6-aminopyridine-3-carbonyl)-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-[1-(1-methylpiperidin-4-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenoxymethyl}pyridine
(2R,6R)-10-methoxy-4-(2-propoxyethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[3-(3-ethylphenoxy)propyl]-N-methyloxane-2-carboxamide
6-methoxy-3-methyl-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1-benzofuran-2-carboxamide
N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
3-[5-(3,3,4,4-tetrafluorobutyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
4-[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[3-(4-tert-butylbenzoyl)piperidine-1-carbonyl]cyclopropan-1-amine
4-(cyclopropylmethyl)-1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-(propan-2-yl)-1,4-diazepan-5-one
3-chloro-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
3-(2-amino-1,3-thiazol-4-yl)-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}propanamide
6-cyclopentyl-N,1-dimethyl-N-(1,2-oxazol-5-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-chloro-6-[3-(2-ethylphenoxy)azetidin-1-yl]pyridine-2-carboxylic acid
1-cyclohexyl-1-[2-(ethylsulfanyl)ethyl]-3-[3-(4H-1,2,4-triazol-4-yl)phenyl]urea
methyl 4-(5-{[(2-methoxyethyl)(propan-2-yl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
1-ethyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)piperidine-4-carboxamide
5-(2-fluorophenyl)-N-[3-(morpholin-4-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
(1R,5S,8S)-3-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-8-methoxy-3-azabicyclo[3.2.1]octane
N-ethyl-2-(3-hydroxyphenyl)-N-[2-(3-methoxyphenoxy)ethyl]acetamide
2-(methoxymethyl)-1-(trimethyl-1H-pyrazole-4-carbonyl)piperidine
(3aR,6aS)-5-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-methoxyethyl)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
6-ethyl-1,5-dimethyl-3-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
(4aR,7aS)-1-[2-(5-oxo-1,4-diazepan-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-(thiophen-2-ylmethyl)acetamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy]-1-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]ethan-1-one
(3aR,7aS)-5-methyl-2-(2-methyl-4-phenylpyridine-3-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-(ethoxymethyl)-N-[1-(pyridin-3-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{[1-(propan-2-yl)-1H-pyrazol-4-yl]formamido}-2-[2-(trifluoromethyl)phenyl]acetic acid
(3R,9aR)-8-[(5-chlorothiophen-2-yl)methyl]-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{4-[(4-ethynylphenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-methyl-N-[(4-phenoxyphenyl)methyl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
N-ethyl-5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-4-methyl-1,3-thiazol-2-amine
3-(3-fluoro-4-methoxybenzoyl)piperidine
4-(2-methoxyphenoxy)-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine
N-{[3-(5-aminopyridin-3-yl)phenyl]methyl}propanamide
[(3R,4S)-1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
3-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]-3,4-dihydro-2H-1λ6,2-benzothiazine-1,1-dione
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
3-[2-(2-fluorophenyl)ethyl]-1-(3-fluoropropyl)piperidine
N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
4-({4-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]piperazin-1-yl}methyl)-1H-indole
3-hydroxy-N-[4-methoxy-3-(methylcarbamoyl)phenyl]-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
2-{4-[(6-fluoroquinolin-2-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
(1S,5R)-6-(cyclopropylmethyl)-3-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-5-chloro-7-methoxy-1-benzofuran-2-carboxamide