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N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(dimethylamino)acetamide
2-[5-(2,3-dihydro-1H-inden-1-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
4-(2-chlorophenoxy)-1-(dimethyl-1,2-oxazole-4-carbonyl)piperidine
N-methyl-4-({5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,3-thiazol-2-amine
2-(7-fluoro-4-methylquinolin-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
methyl (2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[(2-methylpropyl)carbamoyl]pyrrolidine-2-carboxylate
(1S,5R)-3-(5-methyl-1,2-oxazole-3-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,6R)-3-(ethanesulfonyl)-3,9-diazabicyclo[4.2.1]nonane
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
3-[(3R,4S)-1-(1-benzofuran-5-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-4-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}-1,3-oxazole
6-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[(5-methylpyrazin-2-yl)methyl]benzamide
3-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-4-yl}phenol
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-{[(1-methylpiperidin-2-yl)methyl]amino}pyridine-3-carboxamide
2-amino-6-(2,5-dimethylthiophen-3-yl)-4-(3-hydroxyphenyl)pyridine-3-carbonitrile
1-(1,3-benzothiazol-2-yl)-N-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}piperidin-3-amine
1-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
9-(2,6-dimethylpyrimidine-4-carbonyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
6-{[3-(4-methylpiperazin-1-yl)propyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
3-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propanoic acid
methyl 4-{[(4aR,8aS)-1-(4-acetamidobenzoyl)-decahydro-1,6-naphthyridin-6-yl]methyl}benzoate
7-(7-fluoro-4-methylquinolin-2-yl)-4-[(2-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[1-ethyl-8-(1-methoxypropan-2-yl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-4-phenyl-5-(1-propyl-1H-imidazol-2-yl)-1H-imidazole
4-methyl-6-[2-(methylsulfanyl)phenyl]pyrimidin-2-amine
9-(2-hydroxyethyl)-1-methyl-4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-4-(4-methoxyphenoxy)piperidine
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-methoxyphenyl)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
(3R,4S)-1-(4-chloro-2-methylbenzoyl)-4-cyclopropylpyrrolidin-3-amine
6-fluoro-2-({[2-hydroxy-2-(pyridin-2-yl)ethyl]amino}methyl)quinolin-4-ol
N-(4-{1-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1H-imidazol-2-yl}phenyl)acetamide
N-(4-fluorophenyl)-4-{[4-(piperazin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
3-[1-(2-carbamoylphenyl)-1H-pyrazol-4-yl]benzoic acid
N-{1-[1-(3-methoxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
N,2-dimethyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-amine
4-ethyl-5-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1,2,3-thiadiazole
N-[2-(3-fluorophenyl)ethyl]-2-[4-(4-{[2-(pyrazin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
(2S)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(1H-imidazol-2-yl)benzamide
4-(4-cyclopentyl-1,4-diazepan-1-yl)-5-ethylpyrimidin-2-amine
1-[(5-chlorofuran-2-yl)methyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
N-[(3S,4R)-4-(4-methylphenyl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-yl]acetamide
(1S,5R)-3-cyclobutanecarbonyl-6-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
(3R,4R)-1-(1-cyclobutanecarbonylpiperidin-4-yl)-3-cyclopropyl-4-methylpyrrolidin-3-ol