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4-{1-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}pyrimidin-2-amine
N-(2-{1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]piperidin-2-yl}ethyl)acetamide
[(5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}thiophen-3-yl)methyl]dimethylamine
N-[(3R,4S)-1-cycloheptyl-4-cyclopropylpyrrolidin-3-yl]-4-(1H-1,2,4-triazol-1-yl)butanamide
2-{2-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
3-[(4-methoxyphenyl)methyl]-1-methyl-8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{1-[(3-methoxyphenyl)methyl]-5-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
1-[2-(4-propanoylphenoxy)acetyl]imidazolidin-4-one
1-(2-methoxyphenyl)-4-[2-(1-propylpiperidin-4-yl)acetyl]piperazin-2-one
2-[(2-hydroxyethyl)({3-[5-(2-methylphenyl)-4-phenyl-1H-imidazol-1-yl]propyl})amino]ethan-1-ol
N-[2-(4-chlorobenzenesulfonamido)ethyl]-2-(2-oxoazepan-1-yl)acetamide
1-(2-methoxy-5-phenylphenyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
N-benzyl-N-(cyclobutylmethyl)-1-cyclohexyl-1H-1,2,3-triazole-4-carboxamide
1-(2-propoxyacetyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(1R,2R,6S,7S)-4-(2,6-dimethylpyridine-4-carbonyl)-4-azatricyclo[5.2.1.02,6]decane
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(2-phenylethyl)acetamide
8-(3,6-dimethylpyrazin-2-yl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
1-[(3-methylpyridin-2-yl)methyl]-4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
1-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-3-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
ethyl 4-[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]piperidine-1-carboxylate
N-{[5-(2-amino-2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methoxyacetamide
1-(5-acetyl-2-ethoxyphenyl)-3-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]urea
1-(4-methylbenzenesulfonyl)-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazine
4-chloro-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-2-(pyrrolidin-1-yl)-1,3-thiazole
1-(butan-2-yl)-N-(furan-2-ylmethyl)-4-oxo-5-(4-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
methyl 4-{4-[(2R)-2-amino-2-phenylacetyl]piperazin-1-yl}benzoate
2-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidine-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline
methyl 6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-3-carboxylate
N,N-diethyl-1-[1-(quinolin-5-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
[4-({1-[2-(methylsulfanyl)benzoyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-[1-(2,5-difluorophenyl)cyclopropyl]-2,2-dimethyloxane-4-carboxamide
1-ethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-(1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)-1H-1,3-benzodiazole
1-{1-[4-(ethylamino)pyrimidin-2-yl]piperidin-4-yl}piperidin-4-ol
4-{3-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]propoxy}benzamide
5-{[(1-hydroxybutan-2-yl)[(2-methylphenyl)methyl]amino]methyl}-2-methoxyphenol
N-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
ethyl 5-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-1-(4-methoxyphenyl)-1H-pyrazole-4-carboxylate
1-{1-[2-(pyrrolidin-3-yl)benzoyl]piperidin-4-yl}piperidin-4-ol
2-cyclopropyl-N-[3-(2-fluorophenyl)propyl]pyrimidine-5-carboxamide
5-{2-tert-butylimidazo[1,2-a]pyridin-3-yl}pyrimidine
1-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
1-[2-(methylsulfanyl)pyrimidin-4-yl]-N-[2-(pyrazin-2-yl)ethyl]piperidin-4-amine
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)acetamide
1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-2-(pyridin-3-yloxy)ethan-1-one
5-(3-fluorophenyl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1,2,4-triazin-3-amine
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]-4-{[1-(thiophen-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide