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3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}propanamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(1-ethyl-1H-imidazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(propan-2-yl)phenyl]urea
4-(1H-imidazol-1-yl)-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylic acid
3-[4-(6-ethoxy-2,3-dihydro-1H-inden-5-yl)-1H-1,2,3-triazol-1-yl]propane-1,2-diol
2,3,6-trimethyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}quinoline-4-carboxamide
[(3R,4R)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
N-{[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-3-yl]methyl}quinoline-8-sulfonamide
5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-N-methyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-3-carboxamide
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-3,5-dimethyl-1H-pyrazole-4-sulfonamide
2-(2-methoxyethyl)-9-(5-methylpyrazine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(4-{[3-(ethoxymethyl)-1-methyl-1H-1,2,4-triazol-5-yl]methoxy}phenyl)ethan-1-one
1-(azocan-1-yl)-3-[2-methoxy-4-({[2-(pyridin-3-yloxy)ethyl]amino}methyl)phenoxy]propan-2-ol
[(3R,4R)-1-[2-(2-fluorophenyl)benzoyl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
1-[5-methoxy-2-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
6-methoxy-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]hexan-1-one
3-[methyl({2-oxo-2-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl})amino]-1λ6-thiolane-1,1-dione
1-[4-(pyrazin-2-yl)piperazin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
[1-(2-amino-4-methylpyrimidine-5-carbonyl)piperidin-4-yl](pyridin-2-yl)methanol
(2S,4R)-4-amino-N-ethyl-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)pyrrolidine-2-carboxamide
2-{4-[3-(cyclopropylcarbamoyl)piperidin-1-yl]piperidin-1-yl}-N-methylpyridine-3-carboxamide
ethyl[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)sulfamoyl]methylamine
N-(2-fluoroethyl)-3-{[2-(2-methoxyethyl)piperidin-1-yl]sulfonyl}benzamide
N-methyl-N-(thiophen-3-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
7-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(2-oxo-2-{spiro[azepane-4,2'-chromene]-1-yl}ethyl)-1,3-oxazolidin-2-one
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-7-oxo-2-(thiophene-2-amido)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
(1-benzothiophen-2-ylmethyl)(ethyl){[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
1,3-dimethyl-6-(pyridin-4-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-(1H-imidazol-4-yl)ethyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
6-({[(8-methoxyquinolin-5-yl)methyl](methyl)amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-{1H-pyrrolo[2,3-b]pyridin-4-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-(difluoromethyl)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-pyrazole-5-carboxamide
3,5-dimethyl-1-{4-[3-(propoxymethyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazole
3-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]propanamide
(2S,4S)-4-amino-N-(propan-2-yl)-1-[(2,4,5-trimethoxyphenyl)methyl]pyrrolidine-2-carboxamide
methyl 3-(furan-2-amido)-6-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
N4,5,6-trimethyl-N4-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrimidine-2,4-diamine
2-(2-{4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}ethyl)pyridine
5-({4-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)-N-methylfuran-2-carboxamide
N-{2-[bis(propan-2-yl)amino]ethyl}-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
N-methyl-N-(2-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)methanesulfonamide
N-(furan-2-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
(2S,4R)-1-[(4-chlorophenyl)methyl]-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
2-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyrimidine
1-ethyl-4-{[2-(4-methoxy-2,3-dimethylphenyl)-1H-imidazol-1-yl]methyl}pyrrolidin-2-one
(2R,3R)-3-(dimethylamino)-1'-(2-methylbenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-{[3-(2-aminoethyl)phenyl]methyl}-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
5-(2,5-dimethylphenoxymethyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,2-oxazole-3-carboxamide