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(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]piperidin-3-ol
2-methyl-N-(4-{[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]carbamoyl}phenyl)furan-3-carboxamide
(1S,4S)-2-(2-chlorophenyl)-5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
3-{1-cyclopentyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-4-methoxyphenol
N-[(3-fluorophenyl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
4-[(3-phenyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
4-[(3,4-dimethoxyphenyl)methyl]-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
(1R,5S)-3-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-3,8-diazabicyclo[3.2.1]octane
4-chloro-5-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-1-methyl-1H-pyrazole
methyl 5-[4-amino-2-(morpholin-4-yl)-7-oxo-5H,6H,7H,8H-pyrido[2,3-d]pyrimidin-5-yl]-2-hydroxybenzoate
1-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}propan-1-one
2-hydroxy-1-{7-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}propan-1-one
3-{[(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]methyl}benzoic acid
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-[4-(1H-pyrazol-4-yl)butanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-methoxy-1-{2-[3-(morpholine-4-carbonyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
N-[(2S)-1-methoxy-3-phenylpropan-2-yl]-2-(2-oxopiperidin-1-yl)acetamide
3-[5-({8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)thiophen-3-yl]prop-2-yn-1-ol
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chlorophenyl)urea
4-[(dimethylamino)methyl]-1-(4-phenylbenzenesulfonyl)azepan-4-ol
3-{[(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)amino]methyl}-1λ6-thiolane-1,1-dione
3-(1-methyl-1H-pyrazol-4-yl)-1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propan-1-one
4-(2-amino-6-methylpyrimidine-4-carbonyl)-3-(3-fluorophenyl)piperazin-2-one
1-[(4-methoxyphenyl)methyl]-4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperazin-2-one
4-(4-fluorophenyl)-2-({[1-(naphthalen-1-yl)ethyl]amino}methyl)phenol
N-ethyl-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}furan-2-carboxamide
3-[2-(dimethylamino)phenyl]-N,N,1-trimethyl-1H-1,2,4-triazol-5-amine
(3S,4S)-1-[4-(methylcarbamoyl)benzenesulfonyl]-4-propylpyrrolidine-3-carboxylic acid
2-{[(1S,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
2-{4-[(2-methoxyphenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
methyl 4-(4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
7-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-{1-[3-(2-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}pyridine
5-chloro-2-[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
2-(5-chloro-2-ethoxyphenyl)-2-[4-(hydroxymethyl)piperidin-1-yl]acetic acid
2-{[4-(3-chlorophenyl)-5-(piperidin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-methyl-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)-5-sulfamoylbenzamide
{2-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]-1-(2-methylphenyl)ethyl}dimethylamine
1-[5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]-3-phenylpropan-2-ol
N4-{[3-(dimethylamino)thiolan-3-yl]methyl}-N2,N2,5,6-tetramethylpyrimidine-2,4-diamine
1-(2-{[butyl(methyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
5-(4-aminopiperidine-1-carbonyl)-1-cyclohexyl-3-(cyclopropylmethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
(3aR,6aR)-2-benzyl-N-[2-(1H-imidazol-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2,2-dimethyl-4-{[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazol-4-yl]methyl}morpholine
1-{4-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,4-diazepan-1-yl}ethan-1-one
N-cyclohexyl-3-[4-phenyl-5-(trimethyl-1H-pyrazol-4-yl)-1H-imidazol-1-yl]propanamide
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
1-[4-(3-fluorophenyl)phenyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-amine
2-(2-cyclopropylpyrimidin-5-yl)-6,8-dimethyl-4-(morpholine-4-carbonyl)quinoline
N-methyl-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]propanamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]hexane-1,5-dione