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2-(dimethylamino)-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
9-methoxy-10-(thiomorpholine-4-carbonyl)-3-[4-(thiophen-2-yl)butanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-ethyl-3-[2-(5-fluoro-2-methoxyphenyl)-1H-imidazol-1-yl]-2-methylbenzamide
5-(6,7-diethoxy-3-methyl-1-benzofuran-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
(3S,4S)-1-{[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-4-(naphthalen-2-yl)piperidin-3-ol
N4-ethyl-N2-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)pyrimidine-2,4-diamine
N-[(3R,4S)-1-(1,3-dihydroxypropan-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-3-(thiophen-3-yl)propanamide
9-methyl-N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]-9H-carbazole-3-carboxamide
N-(2-methoxyethyl)-4-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-pyrrolo[2,3-b]pyridin-6-amine
4-benzyl-1-methyl-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-[2-(pyridin-2-yl)piperidine-1-carbonyl]-2-(pyridin-4-yl)pyrimidine
5-[2-(morpholin-4-ylmethyl)phenyl]-N-(pyridin-3-yl)furan-2-carboxamide
3-[1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)azetidin-3-yl]pyridine
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-hydroxyacetamide
methyl({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl})[1-(1,2-oxazol-3-yl)ethyl]amine
8-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-(3-chloro-4-methoxyphenyl)-3-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}urea
3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}urea
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
3-cyclohexyl-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
4-{[4-(quinolin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-(2-hydroxyethyl)-2-(2,2,6,6-tetramethylpiperidin-4-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
methyl (2R,4S)-1-[(3-chlorophenyl)methyl]-4-hydroxypiperidine-2-carboxylate
3-(2,3-difluorophenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
2-[(1S,5R)-6-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
(4aS,7aR)-1-[(3-methyl-1-benzofuran-2-yl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(pyrrolidin-3-yl)acetamide
5-{2-oxo-2-[3-(pyridin-4-yl)azetidin-1-yl]ethyl}-3-propylimidazolidine-2,4-dione
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-N-[(2-methoxyphenyl)methyl]-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxamide
7-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)-1,2,3,4-tetrahydroquinoxalin-2-one
5-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1-methyl-1,2-dihydropyridin-2-one
4-(3,4-dimethoxyphenyl)-3-(1-methylpiperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidine-2,4-diamine
2-(1H-indol-3-yl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
2-(1H-indazol-1-yl)-1-{4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
4-{[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-4,4,4-trifluoro-N-(2-hydroxyethyl)butanamide
3-[5-(2,3-difluoro-6-methoxybenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
2-[(1S,5R)-6-[2-(3-chlorophenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N4-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-5-methylpyrimidine-2,4-diamine
1-{4-[2-methoxy-4-(thiomorpholine-4-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
N-[(3-methylpyridin-4-yl)methyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]pyridin-2-amine
N-({5-[(2-fluoro-4-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
4-(3,4-dimethoxybenzoyl)-2-[(3-fluorophenyl)methyl]morpholine
2-oxo-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1,2-dihydroquinoline-4-carboxamide
1-(3-methylpyridin-4-yl)-4-[4-(1H-pyrazol-3-yl)benzoyl]-1,4-diazepane
5-fluoro-N-methyl-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine