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4-[(1-acetylpiperidin-4-yl)oxy]-N-[2-(diethylamino)ethyl]-3-methoxybenzamide
5,6-dimethyl-N-[3-(4-methylpiperazin-1-yl)propyl]pyrimidin-4-amine
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-[(3S,4R)-1-(2-phenyl-1,3-thiazole-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N,3,5-trimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]adamantane-1-carboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperidine
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-phenylethan-1-one
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
N-[2-(dimethylamino)ethyl]-3-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]-N-methylbenzamide
2-[4-(5-ethyl-1,3,4-oxadiazol-2-yl)-1-(furan-3-ylmethyl)piperazin-2-yl]ethan-1-ol
N-(3-hydroxypropyl)-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
{5-[(E)-2-phenylethenyl]-1H-indol-2-yl}methanol
6-cyclopropyl-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}pyrimidin-4-amine
2-(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
3-(2-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-[furan-2-yl(phenyl)methyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
5-chloro-4,6-dimethyl-2-oxo-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,2-dihydropyridine-3-carboxamide
1-[3-(dimethylsulfamoyl)propyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
(3S,4S)-4-(propan-2-yl)-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxylic acid
2-(6-methylpyridine-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethyl-1H-pyrrole-3-carboxamide
4-methoxy-N-[2-(7-{[5-(methoxymethyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
(4aS,7aR)-1-(3-methyl-1H-pyrazole-5-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[2-(4-fluorophenyl)-2-hydroxyacetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(2-methoxyethyl)-1-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(3-fluorophenyl)-2-{4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]morpholin-3-yl}acetamide
ethyl 3-benzyl-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxylate
5-ethyl-2,3-dimethyl-N-[3-(methylsulfanyl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-5-methyl-1,3,4-oxadiazol-2-amine
2-[3-(2-fluorophenoxy)azetidin-1-yl]-5-propyl-1,3,4-oxadiazole
1-benzyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrrolidin-3-amine
(1S,5R)-6-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-propoxybenzamide
3-[methyl({2-[4-(piperidin-1-ylmethyl)piperidin-1-yl]pyrimidin-4-yl})amino]propane-1,2-diol
7-(1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decane
(2S)-3-(1H-imidazol-4-yl)-2-(2-oxo-5,5-diphenylpiperidin-1-yl)propanamide
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
1-(3-fluorophenyl)-N-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
(3S,4S)-4-[4-(2-fluoro-4-methanesulfonylphenyl)piperazin-1-yl]-1-methylpyrrolidin-3-ol
3-chloro-4-{[(1-methylpiperidin-4-yl)(pyridin-3-ylmethyl)amino]methyl}phenol
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}oxolane-3-carboxamide
(2R,3R,6R)-5-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(dimethyl-1,3-thiazol-5-yl)-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]acetamide
4-(4-phenyl-1H-pyrazol-5-yl)-1-(1,2,5-thiadiazole-3-carbonyl)piperidine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-amine
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(2-methyl-1H-pyrrole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidin-3-ol