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N-[(2-chlorophenyl)methyl]-1,3-dimethyl-2,6-dioxo-N-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(3R,5S)-N-(2-methylpropyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
1-[3-(1H-imidazol-2-yl)benzoyl]-4-phenylpiperidine-4-carbonitrile
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-(2-methoxyethyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 3-benzyl-1-[(4-methoxyphenyl)carbamoyl]piperidine-3-carboxylate
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(2-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)acetamide
N-{1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}methanesulfonamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2,4-difluoro-3-methoxybenzamide
N-ethyl-5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)pyrimidin-2-amine
N-tert-butyl-7-[(3-methoxyphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
2,2-dimethyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}propanamide
(1s,4s)-4-(4-{1-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}-1H-1,2,3-triazol-1-yl)cyclohexan-1-amine
2-(4-chloro-3,5-dimethylphenoxy)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]quinoxaline
5-fluoro-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]quinazolin-4-amine
4-(3-methylphenoxy)-1-[2-(pyridin-2-yl)acetyl]piperidine-4-carboxylic acid
4-(2,3-dimethoxy-5-methylphenyl)-N,6-dimethylpyrimidin-2-amine
N-(2H-1,3-benzodioxol-5-yl)-3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carboxamide
1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-5-[1-(ethanesulfonyl)ethyl]-1H-1,2,4-triazole
3-cyclopropyl-5-[2-(difluoromethoxy)phenyl]-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
3-[6-(dimethylamino)pyrimidin-4-yl]benzoic acid
5-ethyl-N-{[3-methyl-7-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1,2-oxazole-3-carboxamide
[1-({1-[(4-methylphenyl)methanesulfonyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
2-(cyclohex-3-en-1-yl)-1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazole
1-[(1,4-dimethyl-1H-pyrazol-5-yl)methyl]-4-(piperidin-1-yl)piperidine-4-carboxamide
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-4-yl)ethyl]amine
(2S,4S)-1-cyclohexyl-N-ethyl-4-[3-(5-methyl-1H-pyrazol-1-yl)propanamido]pyrrolidine-2-carboxamide
(1S,6R)-9-(5-ethyl-1,3-oxazole-4-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
2-(1,2-benzoxazol-3-yl)-N-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]acetamide
3-hydroxy-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1,2-oxazole-5-carboxamide
(4aR,7aS)-1-butanoyl-4-(3-chlorobenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-(1,3-oxazole-5-carbonyl)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-2-carboxamide
1-tert-butyl-N-ethyl-5-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]pyrrolidine-3-carboxamide
(3S,4R)-4-(2-methoxyphenyl)-1-(2-methoxypyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
3-({1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}methyl)benzoic acid
4-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)thiomorpholine
3-({[2-(cyclohex-1-en-1-yl)ethyl]carbamoyl}methyl)-N-cyclopentylmorpholine-4-carboxamide
N-cyclohexyl-3-{[(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]methyl}-N-methylpyridin-2-amine
1-(oxolan-2-ylmethyl)-N-(quinolin-6-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-[3-(dimethylamino)propyl]-8-[(2-fluoro-5-methoxyphenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1,9-dimethyl-4-({4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(2-oxo-2-{4-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-1-yl}ethyl)-2,3-dihydro-1H-isoindol-1-one
N-[(3S,4R)-1-(2,3-dimethyl-1H-indole-5-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
1-[(2,3-difluorophenyl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
9-(2-phenylpropyl)-1,4,9-triazaspiro[5.5]undecan-5-one
(3S,4S)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-(naphthalen-2-yl)piperidin-3-ol
{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(3,4-dimethoxyphenyl)methyl]methylamine
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(thiophen-2-yl)propan-2-yl]urea
(3R,4R)-1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol