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2-{2-[5-(4,5-dimethylthiophen-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyrazine
5-methanesulfonyl-2-methyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]pyrimidin-4-amine
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(1-methylpiperidin-3-yl)propan-1-one
8-methyl-3-{[4-(pyrrolidin-1-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-(1-methylpiperidin-4-yl)-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
N,6-dimethyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
2-chloro-N-[2-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)ethyl]benzamide
9-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
(1S,5R)-6-(2,3-dihydro-1H-indene-5-carbonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-{2-[1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
6-chloro-2-[(4-methanesulfonylphenyl)methyl]-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
1-[(1-{6-[butyl(methyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
N-[5-methoxy-2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-[4-(pyrazin-2-yl)piperazin-1-yl]ethan-1-one
5-{2-azaspiro[4.4]nonane-2-carbonyl}-2-(4-methylphenyl)pyrimidin-4-ol
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)propanamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N,2-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
3-[2-(4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidin-1-yl)-2-oxoethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
[(3R,4R)-1-cycloheptanecarbonyl-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
2-acetyl-8-(4-carboxy-6-methylpyrimidin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-methyl-N-[2-(morpholin-4-yl)ethyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
1-{[2-(2-hydroxyethoxy)phenyl]methyl}-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}thiophene-2-sulfonamide
2-(2-hydroxyethyl)-9-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
4-methyl-2-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
4-ethyl-3-{1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cycloheptyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
2-(naphthalene-2-sulfonyl)-2,8-diazaspiro[4.5]decane
2-(2,4-dioxoimidazolidin-1-yl)-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]acetamide
1-[4-(ethylamino)pyrimidin-2-yl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
2-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)propanamide
2-[(2-chloro-4-fluorophenyl)methyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane
N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
[(3S,5R)-1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-{3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]benzenesulfonyl}-1,4-diazepane
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-methyl-3-(morpholin-4-yl)propan-1-one
N-[(5-chloro-2-methoxyphenyl)methyl]-N,1-dimethyl-3-propyl-1H-pyrazole-5-carboxamide
methyl(oxolan-3-ylmethyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-cyclohexyl-5,6-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[3-(dimethylamino)propyl]-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-{6,8-dioxo-2,7-diazaspiro[4.4]nonan-2-yl}-6-(5-methylthiophen-2-yl)pyridine-3-carboxylic acid
N-(1-methoxypropan-2-yl)-4-(pyridin-2-yl)pyrimidin-2-amine
2-cyclopropyl-9-[4-(4-fluorophenyl)-4-oxobutyl]-2,9-diazaspiro[5.5]undecan-3-one
[1-(2-chlorophenyl)ethyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
3-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}-2-methylpyridine
4-methyl-2-(4-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)pyridine
methyl({pyrazolo[1,5-a]pyrimidin-3-ylmethyl})[1-(thiophen-2-yl)ethyl]amine
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(pyrrolidine-1-carbonyl)-1,4-diazepan-5-one