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2-[(3-fluorophenyl)methyl]-4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]morpholine
N-(2-carbamoylethyl)-3-(2-methyl-1H-indol-1-yl)propanamide
N-[1-(2-methoxyphenyl)ethyl]-N,3,4-trimethyl-5-sulfamoylbenzamide
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-(pyridin-3-ylmethyl)-decahydroisoquinoline
4-{[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)amino]methyl}benzene-1-sulfonamide
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
N-[(2,6-difluoro-3-methylphenyl)methyl]-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-(1-{1-[(2E)-5-methyl-2-(propan-2-yl)hex-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
5,6-dimethyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}thieno[2,3-d]pyrimidin-4-amine
N,N-dimethyl-1-[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-3-amine
[(1,5-dimethyl-1H-indazol-3-yl)methyl][1-(3-methoxyphenyl)propan-2-yl]amine
2-({4-[(4-fluorophenyl)methyl]piperidin-1-yl}methyl)pyridine
6-amino-2-{2-[4-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}pyrimidin-4-ol
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[2-(morpholin-4-yl)ethyl]amine
N'-[2-(dimethylamino)ethyl]-N-(5-methyl-1,2-oxazol-3-yl)-N'-[(5-methylthiophen-2-yl)methyl]ethanediamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(5-methylthiophen-2-yl)methyl](oxolan-2-ylmethyl)amine
3-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-5-(thiophen-2-yl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-[({6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-N,N-dimethylbenzene-1-sulfonamide
(3S,4S)-1-(5,6-dimethoxypyrazine-2-carbonyl)-4-methylpiperidine-3,4-diol
1-(5-ethyl-1,3-oxazole-4-carbonyl)-3-(3-fluorophenoxymethyl)piperidine
N1,N1-dimethyl-N3-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}piperidine-1,3-dicarboxamide
1-(4-benzylpiperazin-1-yl)-3-[1-(3-hydroxypropyl)piperidin-3-yl]propan-1-one
(4aR,7aS)-1-(2-methoxyethyl)-4-(5,6,7,8-tetrahydroquinoline-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-hydroxy-6-methyl-4-(4-methyl-2-oxo-2H-chromen-7-yl)-1,2,3,4-tetrahydroquinolin-2-one
5-{2-[2-(trifluoromethyl)phenyl]acetyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(4aS,7aR)-1-(5-hydroxypyrazine-2-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-ethyl-1-methyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S)-N,N-dimethyl-1-[(2E)-3-phenylprop-2-en-1-yl]azepan-3-amine
2-(7-chloroquinolin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]piperazine
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(2,4-dimethylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
5-(1-methylpyrrolidine-3-carbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-N-[(3-chlorophenyl)methyl]propanamide
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl](methyl)[(3-methylpyridin-4-yl)methyl]amine
N-cyclopropyl-1-(3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propanoyl)piperazine-2-carboxamide
3-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}pyrrolidine
4-methyl-1-{[4-(2-methylpropyl)phenyl]methyl}-1,4-diazepan-5-one
1-(6-chloro-1-methyl-1H-indole-2-carbonyl)-3-(hydroxymethyl)pyrrolidin-3-ol
2-ethoxy-3-(2-methyl-1H-imidazol-4-yl)pyridine
methyl 5-[2-(1H-indazol-3-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
4-(1-ethyl-1H-imidazol-2-yl)-1-(2-phenoxybenzoyl)piperidine
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1-(9H-purin-6-yl)piperidin-4-amine
3-(dimethyl-1,2-oxazol-4-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2H-1,3-benzodioxole-5-carboxamide
2-methyl-6-(1-{5-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl)-3,4-dihydropyrimidin-4-one
3-({4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
methyl 2-(2-oxo-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperazin-1-yl)acetate
1-(azepan-1-yl)-3-(4-{[(2-hydroxyethyl)(methyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
(3aS,6aS)-2-cyclopentyl-5-(1H-indole-5-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid