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1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-propoxypropan-1-one
7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-oxo-4-{3-oxo-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}butanamide
N-methyl-5-({[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)-1,2,4-oxadiazole-3-carboxamide
1-{5-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-4-methylpiperazine
1-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-ethyl-3-{2-[(2S)-4-methyl-2-phenylpiperazin-1-yl]-2-oxoethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
1-{3-[1-(3-methoxypropyl)-1H-imidazol-2-yl]-2,4,6-trimethylphenyl}ethan-1-one
N1,N1,N4-trimethyl-N4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1,4-dicarboxamide
1-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidine-3-carboxamide
3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-N-[(3-methylthiophen-2-yl)methyl]aniline
2-{2-[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethoxy}ethan-1-ol
7-(pyrazine-2-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-[(pyridin-3-ylmethyl)amino]pyridine-3-carboxamide
1-{4-[(diethylamino)methyl]-2-methoxyphenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
4-[4-(furan-2-ylmethyl)piperazin-1-yl]-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]acetamide
(3aR,6aR)-2-acetyl-5-[2-(4-methylpiperidin-1-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[4-(morpholin-4-yl)phenyl]-5-[(propan-2-yl)sulfamoyl]benzoic acid
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[2-(3-methoxyphenyl)azetidin-1-yl]acetamide
5,7-dimethyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-[methyl(propan-2-yl)amino]acetamide
ethyl 4-{5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperazine-1-carboxylate
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-methyl-N-(oxan-4-yl)pyridin-2-amine
2-tert-butyl-5-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1,3,4-oxadiazole
(4aR,7aS)-1-(2-methoxyacetyl)-4-[(2-methyl-1,3-oxazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-(2,3-dimethoxy-5-methylphenyl)pyridin-4-amine
N-cyclopropyl-3-(piperidin-3-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
(1,3-benzothiazol-2-ylmethyl)(methyl){[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}amine
N,N-diethyl-1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
1-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}-3-(pyridin-4-yl)propan-1-one
1-(piperidin-1-yl)-3-(2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenoxy)propan-2-ol
1-{1'-[(2-fluoro-5-methoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
3-[1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)azetidin-3-yl]pyridine
N-{3-[6-amino-5-cyano-4-(5-methylfuran-2-yl)pyridin-2-yl]phenyl}propanamide
1-{[1-(5-chloro-2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-3,3-dimethylurea
3,3-dimethyl-1-[(5-{[4-(2-methylpropyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
3-({4-[4-(2-hydroxyethyl)piperazin-1-yl]piperidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
7-(1,3-benzothiazol-2-yl)-4-(pyridazine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-methyl-N-(2-phenylethyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-5-fluoro-4-(morpholin-4-yl)pyrimidin-2-amine
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-2,3-dihydro-1-benzofuran-5-carboxamide
N-[2-(4-phenylpiperidin-1-yl)ethyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
3-(4-hydroxyphenyl)-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-1H-pyrazole-5-carboxamide
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
cyclopentyl 4-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]carbamoyl}amino)benzoate
5-[2-(2-fluorophenyl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-[4-(6-methylpyridine-2-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
N-(3-hydroxy-2,2-dimethylpropyl)-N-methyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide