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8-[4-(3-hydroxy-3-methylbutyl)benzoyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-({4-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
N-propyl-2-(pyridin-3-yl)benzamide
3-[(3,4-dimethylphenyl)[4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]methyl]pyridine
3-[(4-methoxyphenyl)methyl]-8-(1-methoxypropan-2-yl)-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-3-ol
1-(2,3-dihydro-1H-indene-1-carbonyl)-4-(2,6-dimethylpyridin-4-yl)piperazine
3-(3-hydroxy-1,2-oxazol-5-yl)-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propanamide
2-methyl-8-[2-(piperidin-1-yl)-1,3-thiazole-4-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
1-[1-(1-methylcyclopropyl)propan-2-yl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}amine
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3,5-dimethyl-1,2-oxazole-4-sulfonamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N-[(2,4-dimethoxyphenyl)methyl]-5-methyl-1H-pyrazole-4-carboxamide
ethyl 2-amino-3-cyano-4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-6-carboxylate
5-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}-2-(4-methoxyphenyl)pyrimidine
1-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{1-[3-(furan-2-yl)phenyl]piperidin-4-yl}piperidin-4-amine
4-(2,5-dimethylbenzoyl)-2-(4-methylpentyl)morpholine
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-pentylpiperidine
3-{2-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}-1H-indole
(1R,2R)-2-{3-[(2,6-dichlorophenyl)methyl]-5-methyl-1H-1,2,4-triazol-1-yl}cyclohexan-1-ol
N2-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-N4-methylpyrimidine-2,4-diamine
2-[2-(1H-imidazol-4-yl)ethyl]-9-(1H-pyrazole-4-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 3-[3-(azocan-1-yl)propanamido]propanoate
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}acetamide
1-(4-fluorophenyl)-4-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-yl]piperazine
methyl 5-methyl-4-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}-1,2-oxazole-3-carboxylate
(3R,4R)-1-(dimethyl-1,3-thiazole-5-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-4-(1H-pyrazol-3-yl)benzamide
5-[1-(1H-imidazol-1-yl)ethyl]-3-(thiophen-3-ylmethyl)-1,2,4-oxadiazole
3-(2-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)quinoxalin-2-ol
4-(furan-3-ylmethyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(2R,6S)-4-{[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-2,6-dimethylmorpholine
(4-{[methyl(6-methyl-1,3-benzothiazol-2-yl)amino]methyl}oxan-4-yl)methanol
N-[(4-fluorophenyl)methyl]-3-{1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}propanamide
5-[2-(1-ethylpiperidin-4-yl)acetyl]-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N,N-dimethyl-7-[2-(trifluoromethyl)benzenesulfonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-(cyclohexylmethyl)-7-{[(2,2-dimethyloxan-4-yl)amino]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
ethyl({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})(2-methylprop-2-en-1-yl)amine
N-(4-methoxyphenyl)-1-[2-(pent-4-enamido)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-3-carboxamide
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(oxolane-2-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-{1-[(4-ethoxyphenyl)methyl]-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl}ethan-1-ol
N-[(1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-yl)methyl]pyridine-3-carboxamide
2-{4-[(3,4-difluorophenyl)methyl]-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
methyl 6-{[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}pyridine-2-carboxylate