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2-benzyl-8-(pyridazin-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
4-(dimethyl-1,2-oxazole-4-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
8-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-methyl-1H,2H,5H,6H,7H,8H-[1,3]oxazolo[4,5-g]quinoline-2,6-dione
N-(furan-2-ylmethyl)-N,1-dimethyl-5-({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-benzyl-3-ethyl-1-[2-(1H-pyrazol-4-yl)ethyl]-1,4-diazepan-5-one
N-[2-(dimethylamino)ethyl]-3-fluoro-N-[(2-methylphenyl)methyl]pyridine-4-carboxamide
1-cyclohexyl-3-(2-methylquinolin-5-yl)-1-(pyridin-3-ylmethyl)urea
2,3-dimethyl-6-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]quinoxaline
1-(2-methoxyethyl)-4-({1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)piperidine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-5-(oxolan-2-yl)thiophene-2-carboxamide
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-3-(4-phenylphenyl)propan-1-one
4-(4-benzyl-1H-pyrazol-5-yl)-1-(oxane-4-carbonyl)piperidine
1-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
14-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-methoxy-3-methylbenzamide
2,3,5,6-tetramethyl-N-[2-(pyridin-3-yloxy)propyl]benzamide
2-benzyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,3-benzoxazole-5-carboxamide
6-methyl-2-({[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)pyridin-3-ol
1-[2-(3-chlorophenoxy)propanoyl]-4-(2-methylpropyl)-1,4-diazepan-5-one
N-(2-{3-[3-methyl-7-(pyrazin-2-yl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]-1,2,4-oxadiazol-5-yl}ethyl)acetamide
3-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 3-benzyl-1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]piperidine-3-carboxylate
1-{5-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]thiophen-2-yl}ethan-1-one
ethyl 4-{6-[2-(phenylsulfanyl)acetyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
1-(2-aminoethyl)-N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-4-(methylsulfanyl)benzamide
9-(2-methyloxolane-2-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]cyclopropanesulfonamide
4-(2-methanesulfonylphenyl)-2-methylpyridine
2-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]-4-methoxy-N-(2-methoxyethyl)benzamide
{3-[(1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}pyrrolidin-3-yl)methyl]phenyl}methanol
7-(3-chlorophenyl)-4-[2-(pyridin-2-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-[(diethylamino)methyl]-N-(2-methyl-1-benzofuran-7-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
(1R,3S)-3-(2-hydroxyethoxy)-7-(1-phenylcyclopropanecarbonyl)-7-azaspiro[3.5]nonan-1-ol
N-[3-(4-hydroxyphenyl)propyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-[(2,5-dimethylphenyl)methyl]-3-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
(2S,4S)-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)-4-[(pyridin-3-ylmethyl)amino]pyrrolidine-2-carboxamide
2-[8-(2-hydroxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
N-[1-(furan-2-carbonyl)piperidin-4-yl]-2-methoxyquinoline-4-carboxamide
N-{7-oxo-5-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl}cyclobutanecarboxamide
methyl[1-(pyrazin-2-yl)propan-2-yl]{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
2-(2-{1-[2-(2-methoxyphenyl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
2-(2-ethylphenyl)-2-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}acetic acid
1-[6-hydroxy-4-(6-hydroxypyrimidin-4-yl)-1,4-diazepan-1-yl]-2-phenylethan-1-one
N-[2-(dimethylsulfamoyl)ethyl]-N'-(4-methylphenyl)propanediamide
4-{4-[(2-chloro-6-fluorophenyl)methyl]piperazin-1-yl}-2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
5-ethyl-1'-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{[(5-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}ethan-1-ol
1-{2-[5-(3-hydroxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidin-2-one
3-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-[4-(propylsulfamoyl)phenyl]urea