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3-{1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-3-yl}benzoic acid
2-(4-chlorophenyl)-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidine
1-{4-[4-(1-hydroxycyclopentyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2,2-dimethylpropan-1-one
N-ethyl-2-hydroxy-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-5-(1H-pyrrol-1-yl)benzamide
3-(azepane-1-carbonyl)-N-(furan-2-ylmethyl)-N-methyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N'-cyclopentyl-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}butanediamide
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(3S,4R)-1-(2-methyl-1,8-naphthyridine-3-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
N-(2-methylphenyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-carboxamide
N-[4-(4-{[(3,5-dimethoxyphenyl)methyl]amino}piperidin-1-yl)phenyl]-3-phenylpropanamide
3-(2,5-dioxopyrrolidin-1-yl)-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]benzamide
6-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{2-[2-(ethoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
N-methyl-N-[2-(oxan-4-yl)ethyl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine
N-(4-ethoxy-2-fluorophenyl)-4-hydroxy-4-(pyridin-3-yl)piperidine-1-carboxamide
4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-(3,5-dimethylphenyl)piperazin-2-one
1-(2,3-difluoro-4-methylbenzoyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-[(2,6-dimethylpyridin-3-yl)oxy]-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine-4-carboxylic acid
4-methyl-5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1,2,3-thiadiazole
[(3R,4R)-1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2,3,5,6-tetramethyl-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
1-[(2,3-dimethoxyphenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
7-(2-methylphenyl)-4-[(5-methylthiophen-2-yl)methyl]-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-[(3-methoxyphenyl)methoxy]-4-(2-methyl-1H-1,3-benzodiazole-6-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
2-(5-propylthiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-(furan-2-yl)-2-(4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1H-1,2,3-triazol-1-yl)propanoic acid
3-{[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
3-ethyl-N,1-dimethyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
2-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
2-(butylsulfanyl)-6-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}pyrimidin-4-amine
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]cyclopent-1-ene-1-carboxamide
4-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-N-(1-methyl-1H-pyrazol-5-yl)benzamide
4-(4-{4-[5-phenyl-2-(trifluoromethyl)pyrimidin-4-yl]piperidine-1-carbonyl}phenyl)morpholine
8-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[4-(2-ethylpyrimidine-5-carbonyl)piperazin-1-yl]-2-phenoxyethan-1-one
1-methyl-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine-2-carboxylic acid
(1R,5S)-6-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-6-azabicyclo[3.2.1]octane
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-2-methyl-1,3-benzothiazole-6-sulfonamide
N-benzyl-2-(4-{4-[(2,3-dihydro-1H-inden-2-yl)amino]piperidin-1-yl}phenyl)acetamide
5-{[4-(5-methylfuran-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-N-propylpyrimidin-2-amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(oxan-4-yl)piperidin-4-yl]propanamide
7-(2-methoxyethyl)-2-(5-methylthiophene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-cyclopropanecarbonyl-1'-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(furan-2-yl)-2-({2-methoxy-5H,6H,7H-cyclopenta[b]pyridin-3-yl}formamido)propanoic acid
N-methyl-2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]-N-propylacetamide
1-(cyclohexyloxy)-3-{[1-(9H-purin-6-yl)piperidin-4-yl]amino}propan-2-ol
4-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}pyrimidine