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2-methoxy-5-{[3-(pyridine-2-carbonyl)piperidin-1-yl]methyl}pyridine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methyl-N-(pyridin-3-ylmethyl)acetamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[2-(3-fluorophenyl)piperidin-1-yl]ethan-1-one
N-{[5-({[2-(azepan-1-yl)ethyl](ethyl)amino}methyl)furan-2-yl]methyl}-N-methylmethanesulfonamide
3-benzyl-1-methyl-3-[2-(morpholin-4-yl)-2-oxoethyl]-2,3-dihydro-1H-indol-2-one
methyl 1-{[bis(prop-2-en-1-yl)carbamoyl]methyl}piperidine-4-carboxylate
2-(2-methoxyethyl)-9-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-2,9-diazaspiro[5.5]undecan-3-one
3-(1-methylpiperidin-2-yl)-N-[2-(3-methylthiophen-2-yl)ethyl]propanamide
1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-pyrazole
5-(dimethylamino)-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{3-[(4-fluorophenyl)formamido]propanoyl}piperidine-3-carboxylic acid
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-ethyl-N,2-dimethylpyrimidin-4-amine
3-(1H-imidazol-1-ylmethyl)-1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidine
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
8-fluoro-2-[({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amino)methyl]quinolin-4-ol
3-(1-methyl-1H-pyrazol-4-yl)-1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}propan-1-one
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(pyrimidine-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
{2-[(4-methoxypyrimidin-2-yl)oxy]hex-5-en-1-yl}dimethylamine
1-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazole
2-[2-({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
(2S,4R)-4-cyclobutaneamido-N-ethyl-1-[(3-fluoro-4-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
3-(azocan-1-yl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide
N,2,6-trimethyl-4-oxo-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1,4-dihydropyridine-3-carboxamide
N-cyclopropyl-2-(dimethylamino)-2-(2-methylphenyl)-N-propylacetamide
8-(1-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1S,5R)-3-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]-1-(thiophene-2-carbonyl)piperidine
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N-[3-(dimethylamino)propyl]-5-[(pyridin-3-yloxy)methyl]piperidine-3-carboxamide
2-[4-(hydroxymethyl)phenyl]-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
4-{1-azabicyclo[2.2.2]octan-3-yl}-N-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)piperazine-1-carboxamide
N-cyclopentyl-2-[(furan-2-ylmethyl)(pyridin-2-ylmethyl)amino]propanamide
5-(azepan-1-yl)-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-benzyl-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
3-chloro-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)benzamide
N-{4,6-dimethyl-[1,2]thiazolo[5,4-b]pyridin-3-yl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
methyl 2-(N-methyl-1-{3-[(2-methylpropyl)amino]-5-(pyrrolidine-1-sulfonyl)phenyl}formamido)acetate
4-(cyclohexylmethyl)-3-[(4-methylpiperazin-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
1-methyl-N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}-1H-1,3-benzodiazole-5-carboxamide
N-(3-fluorophenyl)-3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-(4-chlorophenyl)-N-({1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
2-[(2-{[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]amino}ethyl)amino]-6-methyl-3,4-dihydropyrimidin-4-one
6-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-{2-chloro-4-[2-(5-acetamido-1H-1,2,4-triazol-3-yl)acetamido]phenyl}-2,2-dimethylpropanamide
(1R,2S)-1-{2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}-2,3-dihydro-1H-inden-2-ol
3-({[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
ethyl 3-[(4-fluorophenyl)methyl]-1-(4-oxo-3,4-dihydrophthalazine-1-carbonyl)piperidine-3-carboxylate
1-(2-methoxy-4-{[(3-methylbutyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol