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2,6-dihydroxy-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}benzamide
N-cyclopropyl-5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 3-[(3S,4R)-1-[(2,5-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanoate
8-[2-hydroxy-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-{2-[4-(trifluoromethyl)phenyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1H-1,2,3-triazole
2-[benzyl({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})amino]ethan-1-ol
6-[4-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-2,3-dihydropyridazin-3-one
1-[1-(1-benzothiophene-5-carbonyl)pyrrolidin-3-yl]-3,5-dimethyl-1H-pyrazole
N-benzyl-2-[(1R,5R)-3-(dimethylsulfamoyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
2-[4-(benzenesulfonyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
2-[(4-chlorophenyl)methyl]-8-(3-hydroxypropyl)-2,8-diazaspiro[4.5]decan-3-one
2,2-dimethyl-3-{[3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propan-1-ol
2-(4-methoxyphenyl)-N-({1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}methyl)acetamide
N-(2-{4-[(8-methylquinolin-5-yl)methyl]morpholin-2-yl}ethyl)acetamide
N4-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-6-ethyl-5-methylpyrimidine-2,4-diamine
N-[(3S,5S)-1-(3-ethoxypropanoyl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-4-methylpyrimidine-5-carboxamide
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]pyridine-3-carbonitrile
N'-(2-fluoro-5-methylphenyl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]butanediamide
N-benzyl-2-butyl-N,4-dimethyl-3-oxopiperazine-1-sulfonamide
4-[5-(dimethyl-1,2-oxazol-4-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]-1-methylpiperidine
(3R,4S)-3,4-dimethyl-1-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-4-ol
[(dimethyl-1,2-oxazol-4-yl)methyl]({[2-(methoxymethyl)pyrimidin-5-yl]methyl})methylamine
2-(3-hydroxypiperidin-1-yl)-1-[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
1-[2-(dimethylamino)-4-{[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-ethoxyethan-1-one
6-cyclopentyl-N,1-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
4-(2-phenoxybenzoyl)-1,4-oxazepan-6-ol
methyl 5-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]-5-oxopentanoate
2-methyl-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
3-butyl-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-3-(pyridin-4-ylmethyl)urea
5-ethyl-2-({4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
1-{3-[9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}imidazolidin-2-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-[(2-methylphenyl)methoxy]azetidine
1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
3-{3-[cyclohexyl(methyl)amino]propyl}-8-(2-hydroxypropanoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(1-cyclohexylpyrrolidin-2-yl)-N-(1,3-thiazol-2-ylmethyl)thiophene-2-carboxamide
2-(4-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
2-{3-[(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)methyl]-2-methyl-1H-indol-1-yl}acetamide
N,N-dimethyl-5-{1-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}pyrimidin-2-amine
3-chloro-4-({1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-ol
1-[4-(1-benzofuran-2-ylmethyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl]-2-methoxyethan-1-one
N-(2,3-dihydroxypropyl)-N-methyl-1-(piperidin-1-yl)cyclohexane-1-carboxamide
1-(5-propyl-1,3,4-oxadiazole-2-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
7-(4-methoxy-2-methylbenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one