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2-[benzyl(methyl)amino]-N-(1-hydroxypropan-2-yl)-2,3-dihydro-1H-indene-2-carboxamide
1-[(2S,4S)-4-(1H-1,2,3,4-tetrazol-1-yl)-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carbonyl]azepane
1-(3-chlorophenyl)-4-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperazin-2-one
1-(2-methylphenyl)-3-{1-[1-(6-methylpyridine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
2-{1-[1-(2,4-dimethylbenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-amine
(1S,5R)-6-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
5,6-dimethyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-2-methoxy-2-methylpropanamide
N-benzyl-3-(pyrrolidin-1-ylmethyl)aniline
N-[2-(2-fluorophenyl)-1-[1-(quinolin-5-ylmethyl)piperidin-4-yl]ethyl]-N,2-dimethylfuran-3-carboxamide
N-ethyl-N,6-dimethyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
6-cyclopentyl-N,1-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(5S,9aS,9bS)-5-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-[2-(3-methoxyphenyl)ethyl]acetamide
5-[4-(cyclopropylamino)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]-N-methylpyrimidin-2-amine
2-[3-(4-methanesulfonylphenyl)phenoxy]acetamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-[3-(pyridin-2-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-chloro-N-(2-methoxyethyl)-1-methyl-N-(1-methylpiperidin-4-yl)-1H-pyrazole-3-carboxamide
9-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-N-methyl-2-oxo-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,2-dihydropyridine-4-carboxamide
4-(2,4-dichlorophenyl)-3-(pyridin-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-benzothiazole
2-methyl-5-(2-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one
2-[(3S,4R)-3-cyclopropyl-4-methanesulfonamidopyrrolidin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1-oxa-7-azaspiro[3.5]nonane-7-carboxamide
11-{[(2,5-difluorophenyl)methyl]amino}-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-1,4-diazepane-6-carboxylic acid
N-(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N,2-dimethylfuran-3-carboxamide
(1R,9aR)-1-{[(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amino]methyl}-octahydro-1H-quinolizin-1-ol
N,5,6-trimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
[(2-chloro-3,6-difluorophenyl)methyl](methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
1-[(2-methoxyphenyl)methyl]-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
N-[(1-methylpyrrolidin-3-yl)methyl]-3-(thiophen-2-yl)propanamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-propylacetamide
3-butyl-1-methyl-4-(2-phenoxyethanesulfonyl)piperazin-2-one
1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-2-(3-fluorophenoxy)ethan-1-one
(2R,3R)-3-[methyl(2-phenylethyl)amino]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-5-methanesulfonyl-2-methylpyrimidine
3-{[4-(5-fluoropyrimidin-2-yl)piperazin-1-yl]methyl}-7-methylquinolin-2-ol
4-{4-[(4-ethylphenyl)methyl]piperazin-1-yl}-2-(3-methoxypropyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(2-methylpropyl)amino]methyl}piperidin-2-one
(1S,5R)-3-(pyrazin-2-yl)-6-{pyrazolo[1,5-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
(1S,6R)-3-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
1-[3-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-oxopropyl]pyrrolidin-2-one
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-[(3,4-dimethoxyphenyl)methyl]-N-[2-(morpholin-4-yl)ethyl]piperidine-3-carboxamide
2-[3-(2-amino-3-cyano-5,6,7,8-tetrahydroquinolin-4-yl)-1H-indol-1-yl]acetamide
N-[2-(pyrazin-2-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methylacetamide
2-fluoro-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-5-sulfamoylbenzamide