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4-(naphthalen-2-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]-1H-1,2,3-triazole
1-[4-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}sulfonyl)phenyl]ethan-1-one
6-[3-(benzyloxy)piperidin-1-yl]-2-methylpyrimidin-4-amine
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-2-(1H-pyrazol-1-yl)acetamide
6-(1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)pyrimidin-4-ol
3-[(4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-{4-[3-methyl-1-(2-methylphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenoxy}ethan-1-ol
5-[(4-methoxynaphthalen-1-yl)methyl]-5-[3-oxo-3-(3-phenylpiperidin-1-yl)propyl]pyrrolidin-2-one
3-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]acetamide
(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-[2-methyl-4-(pyrrolidine-1-carbonyl)phenyl]-3-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}urea
N-[(2-ethoxy-3-methoxyphenyl)methyl]-N-methyl-4-(1H-pyrazol-3-yl)benzamide
(3R,4R)-4-cyclopropyl-1-[(3,5-dimethyl-1H-indol-2-yl)methyl]-3-methylpiperidin-4-ol
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl][(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
5-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}-3-phenyl-1,2-oxazole
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N,N-dimethyl-4-[4-(4-methylphenyl)-3-oxopiperazine-1-carbonyl]piperidine-1-carboxamide
1-(1,4-dithiepan-6-yl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
(2S)-2-{3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]propanamido}propanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-benzyl-1,3-thiazole-4-carboxamide
2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(methylsulfanyl)ethyl]acetamide
(2S,4S)-4-amino-N-methyl-1-(3-methylpyridine-2-carbonyl)pyrrolidine-2-carboxamide
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine
2-methyl-5-(5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine
1-{4-[(3,4-dimethylphenyl)methyl]-6-hydroxy-1,4-diazepan-1-yl}-2-hydroxyethan-1-one
4-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
1-cyclohexanecarbonyl-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4-methylpentan-1-one
3-oxo-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
2-methoxy-5-[({[4-(methylsulfanyl)phenyl]methyl}(propyl)carbamoyl)amino]benzamide
2-methyl-1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(1H-pyrazol-1-yl)propan-1-one
3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}propan-1-one
5-(2-fluorophenoxymethyl)-N-(isoquinolin-5-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-[2-(cyclohex-1-ene-1-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-1-phenylcyclopropane-1-carboxamide
N-(5-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyridin-2-yl)acetamide
1-ethyl-N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-3,5-dimethyl-1H-pyrazole-4-carboxamide
1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2-(trifluoromethyl)benzamide
N-(2-{5-[(cyclohexylmethyl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2-cyclopentylacetamide
2-[9-(2,5-dimethylbenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
N-[1-(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
3-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyridazine
N-[(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)methyl]acetamide
(benzylsulfamoyl)[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amine
2-methoxy-4-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}pyridine-3-carbonitrile
1'-[(3-hydroxypyrrolidin-3-yl)methyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
(2S,4R)-4-amino-N-methyl-1-[2-(4-methylbenzoyl)benzoyl]pyrrolidine-2-carboxamide