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5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-phenyl-1,2,4-oxadiazole
2,4-dimethyl-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-1,3-oxazole-5-carboxamide
N-methyl-N-[2-(morpholin-4-yl)ethyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
7-(1-benzothiophen-3-yl)-4-(1,4-dioxan-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2,3-dihydro-1H-inden-2-yl)-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-amine
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-1-(propan-2-yl)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
4-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-1-(2-methoxyphenyl)-2,2-dimethylpiperazine
7-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-methoxy-3-[3-(2-methoxyphenoxy)propyl]-N-methylbenzamide
2-(dimethylamino)-N-methyl-2-(4-methylphenyl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
2-(1-ethylpiperidin-4-yl)-N-[2-hydroxy-2-(pyridin-3-yl)ethyl]acetamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(trifluoromethyl)benzamide
(4aS,8aR)-6-(1H-pyrazole-3-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-(3,4-difluorophenyl)-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-amine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
benzyl({[(2R)-1-(benzyloxy)-3-hydroxypropan-2-yl]sulfamoyl})amine
N-[2-(benzylsulfanyl)ethyl]-1-(4-fluorophenyl)-2,2-dimethylcyclopropane-1-carboxamide
[5-methyl-7-(2-methyl-1H-imidazol-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)butanamide
3-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]quinoline
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-3-(propan-2-yl)-N-(pyridin-2-ylmethyl)-1,2-oxazole-5-carboxamide
2-ethyl-5-({4-[2-(furan-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)-1,3,4-thiadiazole
7-(1,3-benzothiazol-2-yl)-4-[2-(dimethylamino)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-4-(pyrimidin-2-yloxy)piperidine-1-carboxamide
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-3-(furan-2-yl)propanamide
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}[2-(1H-indol-3-yl)ethyl]amine
4-{8-[2-(dimethylamino)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-methoxypyridine-3-carbonitrile
2-(4-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}phenoxy)pyrimidine
8-(dimethyl-1,3-oxazole-4-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazol-4-yl)ethan-1-ol
2-[4-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)phenyl]-6-(2-methoxyethyl)-3,4-dihydropyrimidin-4-one
1-(2-{[(4-methoxy-2,3-dimethylphenyl)methyl](methyl)amino}ethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(1S)-1-phenylethyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
3-(1H-1,3-benzodiazol-2-yl)-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
2-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,2-benzothiazol-3-one
3-{5-[2-(diethylamino)ethyl]-1,3,4-thiadiazol-2-yl}-1-(2,3-dihydro-1H-inden-1-yl)urea
3-[benzyl({[3-(cyclopentyloxy)phenyl]carbamoyl})amino]propanamide
3-[2-(2-methylphenyl)ethyl]-1-(oxane-4-carbonyl)piperidine
6-methoxy-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrimidin-4-amine
1-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)cyclopropane-1-carboxamide
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
diethyl({[3-(4-propylpiperazine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
7-[(2S)-2-amino-3,3-dimethylbutanoyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
3-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)-N-(4-methylpyridin-3-yl)benzamide
3-(2-ethyl-1H-imidazol-1-yl)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
1-[(1-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}cyclopropyl)methyl]-1H-pyrazole
5-{2-[2,2-bis(prop-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}-1,3-dimethylimidazolidine-2,4-dione
4-(8-chloroquinolin-2-yl)piperazine-2-carboxylic acid