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N,N-diethyl-1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
4-[2-(1,4-oxazepan-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]pyridine-2-carboxylic acid
N-[(3R,4R)-1-[(2-ethylphenyl)methyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
1-(4-{[(cyclohexylmethyl)amino]methyl}-2-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
1-[(3-cyclopentyl-1,2,4-oxadiazol-5-yl)methyl]azepan-2-one
ethyl 1-[6-(1-benzothiophen-3-yl)-3-[(1,2-oxazol-3-ylmethyl)carbamoyl]pyridin-2-yl]piperidine-3-carboxylate
N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-4-(piperidin-3-yl)benzamide
methyl 1-(3-{3-[(benzylamino)methyl]phenoxy}-2-hydroxypropyl)piperidine-4-carboxylate
N-{[2-(4-acetylpiperazin-1-yl)-7-methylquinolin-3-yl]methyl}-N-cyclopropyl-1,3-thiazole-5-carboxamide
1-(2-methoxyphenyl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-pyrazole-4-carboxamide
3-(1H-imidazol-2-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
2-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
2-[3-(4-tert-butylbenzoyl)piperidin-1-yl]ethan-1-ol
4-(3-methoxypropyl)-N-[3-methyl-1-(2-methylpropyl)-1H-pyrazol-5-yl]piperazine-1-carboxamide
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-phenyl-1H-pyrazole-4-carboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-3-(furan-2-yl)propanamide
N-(2-hydroxyethyl)-3-(1H-imidazol-2-yl)-N-[(2-methoxyphenyl)methyl]benzamide
1-{2-[1-(piperidin-3-yl)piperidin-4-yl]ethyl}pyrrolidin-2-one
N-[2-(azepan-1-yl)ethyl]-2-(ethanesulfonyl)-N-(propan-2-yl)propanamide
2-phenyl-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-(2-methoxyethyl)piperazine
(3S,4S)-1-(2-phenylethyl)-4-(piperidin-1-yl)pyrrolidin-3-ol
2-{4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-1-(piperidin-1-yl)ethan-1-one
3-benzyl-4-[3-(1H-pyrazol-4-yl)benzoyl]piperazin-2-one
methyl 3-[(3S,4R)-1-[(3-ethoxy-4-hydroxyphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoate
N-cyclopropyl-1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}piperidine-3-carboxamide
N-[4-(furan-2-yl)phenyl]-1-(thiophen-3-ylmethyl)piperidine-3-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
4-(1,2,3,4-tetrahydroisoquinolin-5-yl)-8-(trifluoromethyl)quinoline
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-4-(piperidine-1-carbonyl)pyridin-2-amine
2-benzyl-9-[(2,3-difluoro-4-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
6-[(dimethylamino)methyl]-N-(4-methoxy-2-methylphenyl)-1,4-oxazepane-4-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-4H-chromen-4-one
4-methyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-1,3-oxazole-5-carboxamide
[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
2-ethyl-6-methyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-4-oxo-1-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-({3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}methyl)benzonitrile
3-{3-ethyl-5-[2-(4H-1,2,4-triazol-4-yl)pyridin-4-yl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
(2S,4S)-4-amino-N-ethyl-1-[(5-ethylpyridin-2-yl)methyl]pyrrolidine-2-carboxamide
8-[(3-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[benzyl(methyl)amino]-3-[4-({[2-(pyridin-3-yloxy)ethyl]amino}methyl)phenoxy]propan-2-ol
(3R,4R)-4-(azepan-1-yl)-1-[(4-methoxynaphthalen-1-yl)methyl]piperidin-3-ol
[(2-cyclohexylpyrimidin-5-yl)methyl](oxolan-2-ylmethyl)propylamine
1-(furan-2-ylmethyl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]piperidine-4-carboxamide
(3S,4S)-4-methyl-1-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)piperidine-3,4-diol
3-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
(4aS,8aR)-6-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-[(3S)-1-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-yl]acetamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(3S)-2-oxoazepan-3-yl]benzamide