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2-(4-methylpentyl)-4-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]morpholine
3-{[1-(6-methylpyridin-2-yl)-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
1-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}-2-[(2-methylphenyl)amino]ethan-1-one
1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-2-(methylamino)-1,3-thiazole-4-carboxamide
4-{[5-(2-methylpropyl)-4-phenyl-1H-imidazol-1-yl]methyl}pyridine
2-benzyl-8-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-2,8-diazaspiro[4.5]decan-3-one
methyl({[5-(oxan-2-yl)furan-2-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
N-(oxolan-2-ylmethyl)-4-[({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}carbamoyl)amino]benzamide
3-(2-amino-1,3-thiazol-4-yl)-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]propanamide
9-(benzenesulfonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetamido]-N-(3-methoxyphenyl)benzamide
4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-cyclopropanecarbonylpiperidine
(3S,4S)-4-cyclopropyl-1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]pyrrolidine-3-carboxylic acid
methyl 4-[(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)carbamoyl]butanoate
5-{[2-(9H-fluoren-2-yl)-1H-imidazol-1-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
(1S,4S)-5-(1-benzylpiperidin-4-yl)-2-(2,5-dimethoxyphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
6-[2-(1-ethylpiperidin-3-yl)-1H-imidazol-1-yl]-2-methyl-1,3-benzothiazole
4-{2-[1-(2-chloro-6-fluoro-3-methylbenzoyl)piperidin-2-yl]ethyl}morpholine
3-chloro-6-methyl-N-(2,2,2-trifluoroethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-[4-(cyclopropylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
1-[(2-methoxyphenyl)methyl]-5-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]piperidin-2-one
3-{[4-(2-amino-5-ethyl-6-methylpyrimidin-4-yl)piperazin-1-yl]methyl}benzonitrile
methyl 2-{3-oxo-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-8-yl}propanoate
1-{2-oxo-2-[4-(thian-4-yl)piperazin-1-yl]ethyl}-1,2-dihydropyridin-2-one
2-(2-chlorophenyl)-N-cyclopropyl-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-{[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzoic acid
4-(1H-imidazol-2-yl)-1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-1,2,3-triazole
1-(pyridin-2-ylmethyl)-4-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
2-(1H-1,2,3,4-tetrazol-5-yl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)acetamide
2-(morpholin-4-yl)-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]pyridine-3-carboxamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(piperidin-3-ylmethyl)benzamide
6-[(piperidin-4-yl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N-[(2-aminopyridin-3-yl)methyl]-6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[4-(cyclobutylamino)-2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-hydroxyethan-1-one
2-hydroxy-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
1-[2-(4-fluorophenyl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(2S,4S)-4-amino-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-N-ethylpyrrolidine-2-carboxamide
5-[2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]thiophene-2-sulfonamide
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-2-methyl-N-[(3S)-2-oxoazepan-3-yl]propanamide
(1S,6R)-9-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[2-(pyrrolidin-1-yl)ethyl]amino}methyl)piperidin-2-one
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]bis(1,3-oxazol-4-ylmethyl)amine
N-[2-(5-methylfuran-2-yl)phenyl]-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carboxamide
N-[(2-propyl-1,3-thiazol-4-yl)methyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(ethoxymethyl)-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidine
2-chloro-5-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl]carbamoyl}amino)-N-ethylbenzamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2,3-dihydro-1-benzofuran-7-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetamide